Affinity DataKi: <1nM ΔG°: <-50.9kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nM ΔG°: -49.6kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nM ΔG°: -49.3kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -47.5kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nM ΔG°: -47.0kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 5.80nM ΔG°: -46.5kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 6.60nM ΔG°: -46.2kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 9.80nM ΔG°: -45.3kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -43.5kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 48nM ΔG°: -41.4kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 62nM ΔG°: -40.7kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 84nM ΔG°: -40.0kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 108nM ΔG°: -39.4kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 169nM ΔG°: -38.3kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 169nM ΔG°: -38.3kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 287nM ΔG°: -37.0kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60.6nMAssay Description:Antagonist activity at androgen receptor in human LNAR cells expressing ARE-PSA-LUC by luminescence analysis in presence of R1881More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Antagonist activity at androgen receptor expressed in human LNAR cells assessed as inhibition of R1881-induced luciferase activity by spectrophotomet...More data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Antagonist activity at androgen receptor expressed in human LNAR cells assessed as inhibition of R1881-induced luciferase activity by spectrophotomet...More data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Antagonist activity at androgen receptor expressed in human LNAR cells assessed as inhibition of R1881-induced luciferase activity by spectrophotomet...More data for this Ligand-Target Pair
Affinity DataIC50: 79.6nMAssay Description:Antagonist activity at androgen receptor in human LNAR cells expressing ARE-PSA-LUC by luminescence analysis in presence of R1881More data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Antagonist activity at androgen receptor expressed in human LNAR cells assessed as inhibition of R1881-induced luciferase activity by spectrophotomet...More data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Antagonist activity at androgen receptor in human LNAR cells expressing ARE-PSA-LUC by luminescence analysis in presence of R1881More data for this Ligand-Target Pair
Affinity DataIC50: 131nMAssay Description:Antagonist activity at androgen receptor expressed in human LNAR cells assessed as inhibition of R1881-induced luciferase activity by spectrophotomet...More data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 144nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 161nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 163nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 165nMAssay Description:Antagonist activity at androgen receptor in human LNAR cells expressing ARE-PSA-LUC by luminescence analysis in presence of R1881More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Antagonist activity at androgen receptor in human LNAR cells expressing ARE-PSA-LUC by luminescence analysis in presence of R1881More data for this Ligand-Target Pair
Affinity DataIC50: 174nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 175nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 178nMAssay Description:Antagonist activity at androgen receptor in human LNAR cells expressing ARE-PSA-LUC by luminescence analysis in presence of R1881More data for this Ligand-Target Pair
Affinity DataIC50: 189nMAssay Description:Antagonist activity at androgen receptor in human LNAR cells expressing ARE-PSA-LUC by luminescence analysis in presence of R1881More data for this Ligand-Target Pair
Affinity DataIC50: 197nMAssay Description:Antagonist activity at androgen receptor in human LNAR cells expressing ARE-PSA-LUC by luminescence analysis in presence of R1881More data for this Ligand-Target Pair
Affinity DataIC50: 263nMAssay Description:Antagonist activity at androgen receptor expressed in human LNAR cells assessed as inhibition of R1881-induced luciferase activity by spectrophotomet...More data for this Ligand-Target Pair