Found 198 with Last Name = 'fillgrove' and Initial = 'kl' 
Affinity DataKi: 540nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Positive allosteric modulation of 5-HT2B receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Positive allosteric modulation of platelet-activating factor receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:In vitro Oxytocin receptor antagonistic activity against rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory activity against bovine cathepsin DMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory activity against aspartic proteinases pepsin from porcineMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:In vitro Oxytocin receptor antagonistic activity against rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 224nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 338nMAssay Description:ETA receptor antagonist activity was measured by inhibition of ET-1 induced vasoconstriction in isolated porcine coronary arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 585nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:In vitro Oxytocin receptor antagonistic activity against rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 2.47E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 4.21E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+3nMAssay Description:In vitro Oxytocin receptor antagonistic activity against rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.47E+3nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Compound was evaluated for the inhibition of microsomal 2,3-oxidosqualene-lanosterol cyclase in Candida albicans microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >2.80E+4nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: >2.80E+4nMAssay Description:In vitro Oxytocin receptor antagonistic activity against rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.80E+4nMAssay Description:In vitro inhibitory potency against human kidney renin.More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Choline AcetyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
