TargetCannabinoid receptor 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]CP-55940 human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 8.90nMAssay Description:Displacement of [3H]CP-55940 human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of rat CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Displacement of [3H]CP-55940 human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Displacement of [3H]CP-55940 human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Displacement of [3H]CP-55940 human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]CP-55940 human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: <631nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Displacement of [3H]CP-55940 human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: <794nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to dopamine 2 receptorMore data for this Ligand-Target Pair