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Found 103 with Last Name = 'fitch' and Initial = 'kj'
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282359(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50:  0.800nMAssay Description:In vitro binding affinity of the compound evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II re...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282358(CHEMBL432734 | N-[4'-(2-Ethyl-6,8-dimethyl-imidazo...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity of the compound evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II re...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284439(CHEMBL15729 | [2-Allyl-6-chloro-4-(2-ethyl-5,7-dim...)
Affinity DataIC50:  2.20nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284453(CHEMBL15517 | [2-Chloro-4-(2-ethyl-5,7-dimethyl-im...)
Affinity DataIC50:  3.40nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285344(CHEMBL40585 | [4-(7-Methyl-2-propyl-imidazo[4,5-b]...)
Affinity DataIC50:  5nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282360(2-Ethyl-6,8-dimethyl-3-[2'-(2H-tetrazol-5-yl)-biph...)
Affinity DataIC50:  5.70nMAssay Description:In vitro binding affinity of the compound evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II re...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284454(CHEMBL15606 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  6nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284445((2-Chloro-phenyl)-[4-(2-ethyl-5,7-dimethyl-imidazo...)
Affinity DataIC50:  8nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284451(CHEMBL279103 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,...)
Affinity DataIC50:  9.5nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282359(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50: >10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284456((2-Chloro-phenyl)-[4-(2-ethyl-5,7-dimethyl-imidazo...)
Affinity DataIC50:  10nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282361(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50: >10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282358(CHEMBL432734 | N-[4'-(2-Ethyl-6,8-dimethyl-imidazo...)
Affinity DataIC50: >10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282360(2-Ethyl-6,8-dimethyl-3-[2'-(2H-tetrazol-5-yl)-biph...)
Affinity DataIC50: >10nMAssay Description:In vitro binding affinity at AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from rat brain memb...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284444(CHEMBL15689 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  11nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284464(CHEMBL15788 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  11nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284460(CHEMBL278983 | [2-Ethyl-4-(2-ethyl-5,7-dimethyl-im...)
Affinity DataIC50:  12nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284465(CHEMBL15847 | [2-Butyl-4-(2-ethyl-5,7-dimethyl-imi...)
Affinity DataIC50:  12nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284463(CHEMBL15730 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  14nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284441(CHEMBL15850 | [2-Chloro-4-(2-ethyl-5,7-dimethyl-im...)
Affinity DataIC50:  15nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284455(CHEMBL15669 | [2-Chloro-4-(2-ethyl-5,7-dimethyl-im...)
Affinity DataIC50:  16nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285349((2-Chloro-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50:  16nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285356((2-Ethoxy-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50:  18nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284462(CHEMBL278234 | [2-Allyl-4-(2-ethyl-5,7-dimethyl-im...)
Affinity DataIC50:  20nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285353((2,6-Dichloro-phenyl)-[4-(7-methyl-2-propyl-imidaz...)
Affinity DataIC50:  21nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284448(CHEMBL280290 | [2,6-Dichloro-4-(2-ethyl-5,7-dimeth...)
Affinity DataIC50:  21nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285345((4-Chloro-2-cyclohexyl-phenoxy)-(4-chloro-phenyl)-...)
Affinity DataIC50:  21nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285349((2-Chloro-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50:  22nMAssay Description:Tested in vitro for Angiotensin II receptor, type 2 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50117909(CHEMBL278176 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284457(CHEMBL15671 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  29nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284442(CHEMBL15882 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  30nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285346(CHEMBL288222 | [4-(7-Methyl-2-propyl-imidazo[4,5-b...)
Affinity DataIC50:  36nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284470(Benzo[1,3]dioxol-5-yl-[4-(2-ethyl-5,7-dimethyl-imi...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285358((2-Methoxy-phenyl)-[4-(7-methyl-2-propyl-imidazo[4...)
Affinity DataIC50:  38nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284459(CHEMBL274260 | [4-(7-Methyl-2-propyl-imidazo[4,5-b...)
Affinity DataIC50:  42nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284444(CHEMBL15689 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  47nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rat midbrain membrane (AT2 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284450(CHEMBL15774 | [2-tert-Butyl-4-(2-ethyl-5,7-dimethy...)
Affinity DataIC50:  50nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285351(CHEMBL39124 | [4-(7-Methyl-2-propyl-imidazo[4,5-b]...)
Affinity DataIC50:  57nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50117909(CHEMBL278176 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284440(CHEMBL278061 | [2-Benzoyl-4-(2-ethyl-5,7-dimethyl-...)
Affinity DataIC50:  60nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rat midbrain membrane (AT2 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285355((3-Chloro-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50:  60nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284461(CHEMBL278955 | [2-Acetyl-4-(2-ethyl-5,7-dimethyl-i...)
Affinity DataIC50:  62nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284459(CHEMBL274260 | [4-(7-Methyl-2-propyl-imidazo[4,5-b...)
Affinity DataIC50:  65nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284443(CHEMBL280456 | [4-(2-Ethyl-6,8-dimethyl-imidazo[1,...)
Affinity DataIC50:  69nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284468(5-Isobutyl-thiophene-2-sulfonic acid {2-benzo[1,3]...)
Affinity DataIC50:  75nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285350(7-Methyl-3-{4-[phenyl-(1H-tetrazol-5-yl)-methoxy]-...)
Affinity DataIC50:  77nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50285347((2-Hexyloxy-phenyl)-[4-(7-methyl-2-propyl-imidazo[...)
Affinity DataIC50:  80nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282361(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50:  83nMAssay Description:In vitro binding affinity of the compound evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II re...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284468(5-Isobutyl-thiophene-2-sulfonic acid {2-benzo[1,3]...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284447(CHEMBL15670 | [4-(2-Butyl-benzoimidazol-1-ylmethyl...)
Affinity DataIC50:  93nMAssay Description:Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rabbit aortic membrane (AT1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
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