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Found 665 with Last Name = 'fossetta' and Initial = 'j'
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227000(3-[4-((R)-1-furan-2-yl-2,2-dimethyl-propylamino)-1...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227005(3-{4-[(R)-1-(4,5-dimethyl-furan-2-yl)-2-methyl-pro...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50226999(2-hydroxy-N,N-dimethyl-3-{4-[(R)-1-(5-methyl-furan...)
Affinity DataKi:  3nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50226995(3-[4-((R)-2,2-dimethyl-1-phenyl-propylamino)-1-oxo...)
Affinity DataKi:  4nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227003(3-[4-((R)-1-benzo[1,3]dioxol-5-yl-2,2-dimethyl-pro...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227001(3-{4-[(R)-2,2-dimethyl-1-(5-methyl-furan-2-yl)-pro...)
Affinity DataKi:  5nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50226996(2-hydroxy-N,N-dimethyl-3-[1-oxo-4-((R)-1-phenyl-pr...)
Affinity DataKi:  5nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248084((R)-2-hydroxy-N,N-dimethyl-3-(4-(1-(5-methylfuran-...)
Affinity DataKi:  7.5nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227010(3-{4-[(R)-1-(3-fluoro-phenyl)-2-methyl-propylamino...)
Affinity DataKi:  8nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227013(2-hydroxy-N,N-dimethyl-3-{4-[(R)-1-(4-methyl-3,4-d...)
Affinity DataKi:  9nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227011(3-{4-[(R)-1-(5-chloro-furan-2-yl)-2,2-dimethyl-pro...)
Affinity DataKi:  9nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50226993(2-hydroxy-3-{4-[(R)-1-(4-isopropyl-furan-2-yl)-pro...)
Affinity DataKi:  9nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50226997(3-{4-[(R)-1-(3-fluoro-phenyl)-2-methyl-propylamino...)
Affinity DataKi:  11nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227006(3-[4-((R)-1-furan-2-yl-2,2-dimethyl-propylamino)-1...)
Affinity DataKi:  11nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227009(3-(4-{[(R)-furan-2-yl-(1-methyl-cyclopropyl)-methy...)
Affinity DataKi:  12nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248113((R)-N-(2-cyanoethyl)-3-(4-(2,2-dimethyl-1-(5-methy...)
Affinity DataKi:  13nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50247950((R)-2-hydroxy-N,N-dimethyl-3-(4-(1-(5-methylfuran-...)
Affinity DataKi:  13nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248115((R)-N-(2-cyanoethyl)-3-(4-(1-(furan-2-yl)-2,2-dime...)
Affinity DataKi:  14nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248038((R)-3-(4-(2,2-dimethyl-1-(5-methylfuran-2-yl)propy...)
Affinity DataKi:  14nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248082((R)-2-hydroxy-N,N-dimethyl-3-(4-(2-methyl-1-(5-met...)
Affinity DataKi:  14nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227004(3-{4-[(benzo[1,3]dioxol-5-ylmethyl)-amino]-1-oxo-1...)
Affinity DataKi:  15nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248037((R)-2-hydroxy-N,N-dimethyl-3-(4-(2-methyl-1-(5-met...)
Affinity DataKi:  15nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248039((R)-3-(4-(1-(furan-2-yl)-2,2-dimethylpropylamino)-...)
Affinity DataKi:  15nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248591((R)-3-(4-(cyclopropyl(phenyl)methylamino)-1,2,5-th...)
Affinity DataKi:  16nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227002(3-[4-((R)-1-furan-2-yl-2,2-dimethyl-butylamino)-1,...)
Affinity DataKi:  16nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248083((R)-(3-(4-(2,2-dimethyl-1-(5-methylfuran-2-yl)prop...)
Affinity DataKi:  18nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248590((R)-3-(4-(1-(3,5-difluorophenyl)propylamino)-1,2,5...)
Affinity DataKi:  20nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM22202(S1P | [32P]S1P | [33P]S1P | sphingosine-1-phosphat...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248547((R)-2-hydroxy-N,N-dimethyl-3-(4-(1-phenylpropylami...)
Affinity DataKi:  21nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227000(3-[4-((R)-1-furan-2-yl-2,2-dimethyl-propylamino)-1...)
Affinity DataKi:  21nMAssay Description:Binding affinity to CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227008(3-{4-[(R)-1-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-2,...)
Affinity DataKi:  24nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM22202(S1P | [32P]S1P | [33P]S1P | sphingosine-1-phosphat...)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM22202(S1P | [32P]S1P | [33P]S1P | sphingosine-1-phosphat...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM22202(S1P | [32P]S1P | [33P]S1P | sphingosine-1-phosphat...)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM22202(S1P | [32P]S1P | [33P]S1P | sphingosine-1-phosphat...)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM22202(S1P | [32P]S1P | [33P]S1P | sphingosine-1-phosphat...)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248114((R)-N-(2-cyanoethyl)-2-hydroxy-3-(4-(1-(4-isopropy...)
Affinity DataKi:  34nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50247972((R)-2-hydroxy-N,N-dimethyl-3-(4-(1-(4-methylfuran-...)
Affinity DataKi:  35nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248589(2-hydroxy-N,N-dimethyl-3-(4-(2,2,2-trifluoro-1-phe...)
Affinity DataKi:  36nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227001(3-{4-[(R)-2,2-dimethyl-1-(5-methyl-furan-2-yl)-pro...)
Affinity DataKi:  38nMAssay Description:Binding affinity to CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248112((R)-3-(4-(2,2-dimethyl-1-(5-methylfuran-2-yl)propy...)
Affinity DataKi:  38nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248546((S)-3-(4-(3,3-dimethylbutan-2-ylamino)-1,2,5-thiad...)
Affinity DataKi:  43nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248115((R)-N-(2-cyanoethyl)-3-(4-(1-(furan-2-yl)-2,2-dime...)
Affinity DataKi:  44nMAssay Description:Displacement of IL8 from CXCR2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248592((R)-3-(4-(1-(2,3-dihydro-1H-inden-5-yl)-2,2-dimeth...)
Affinity DataKi:  44nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227003(3-[4-((R)-1-benzo[1,3]dioxol-5-yl-2,2-dimethyl-pro...)
Affinity DataKi:  46nMAssay Description:Binding affinity to CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227005(3-{4-[(R)-1-(4,5-dimethyl-furan-2-yl)-2-methyl-pro...)
Affinity DataKi:  50nMAssay Description:Binding affinity to CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50247947((R)-3-(4-(1-(benzo[d][1,3]dioxol-5-yl)-2,2-dimethy...)
Affinity DataKi:  52nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50248036((S)-2-hydroxy-N,N-dimethyl-3-(4-(2,2,2-trifluoro-1...)
Affinity DataKi:  53nMAssay Description:Displacement of IL8 from CXCR1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227007(2-hydroxy-N,N-dimethyl-3-[1-oxo-4-((S)-1,2,2-trime...)
Affinity DataKi:  58nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50227006(3-[4-((R)-1-furan-2-yl-2,2-dimethyl-propylamino)-1...)
Affinity DataKi:  61nMAssay Description:Binding affinity to CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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