Affinity DataKi: 0.0880nM ΔG°: -59.7kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 0.160nM ΔG°: -58.2kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 0.290nM ΔG°: -56.6kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 0.330nM ΔG°: -56.3kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 0.740nM ΔG°: -54.2kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nM ΔG°: -52.6kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 2.24nM ΔG°: -51.4kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 5.14nM ΔG°: -49.2kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 8.91nM ΔG°: -47.8kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 21.7nM ΔG°: -45.5kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataKi: 24.9nM ΔG°: -45.1kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
Affinity DataIC50: 0.640nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 0.720nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair