Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
Dainippon Pharmaceutical
Curated by PDSP Ki Database
Dainippon Pharmaceutical
Curated by PDSP Ki Database
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PIM1 (unknown origin) by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibition of GSK3beta (unknown origin) by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetLanosterol synthase(Homo sapiens (Human))
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human C-terminal His6-tagged OSC expressed in Pichia pastoris GS115 using 2,3-oxidosqualene as substrate after 90 mins by 1H NMR methodMore data for this Ligand-Target Pair
TargetDeath-associated protein kinase 1(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of DAPK1 (unknown origin) by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetLanosterol synthase(Homo sapiens (Human))
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human C-terminal His6-tagged OSC expressed in Pichia pastoris GS115 using 2,3-oxidosqualene as substrate after 90 mins by 1H NMR methodMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetTrypanothione synthetase(Trypanosoma cruzi)
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of Trypanosoma cruzi strain CL Brener N-terminal poly-His tagged spermidine synthase expressed in Escherichia coli BL21(DE3) using 50 uM p...More data for this Ligand-Target Pair
TargetLanosterol synthase(Homo sapiens (Human))
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human C-terminal His6-tagged OSC expressed in Pichia pastoris GS115 using 2,3-oxidosqualene as substrate after 90 mins by 1H NMR methodMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetLanosterol synthase(Homo sapiens (Human))
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of human C-terminal His6-tagged OSC expressed in Pichia pastoris GS115 using 2,3-oxidosqualene as substrate after 90 mins by 1H NMR methodMore data for this Ligand-Target Pair
TargetTrypanothione synthetase(Trypanosoma cruzi)
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Inhibition of Trypanosoma cruzi strain CL Brener N-terminal poly-His tagged spermidine synthase expressed in Escherichia coli BL21(DE3) using 0.5 mM ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PIM2 (unknown origin) by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetSpermidine synthase(Sus scrofa)
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of porcine spermidine synthase assessed as production of labeled 5'-methylthioadenosine using putrescine as substrate by enzymatic assay i...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of PIM3 (unknown origin) using FL-Peptide 1 (5-FAM-AKRRRLSSLRA-COOH) substrate incubated for 2 hrs by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
TargetTrypanothione synthetase(Trypanosoma cruzi)
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
National Institute Of Advanced Industrial Science And Technology (Aist)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi strain CL Brener N-terminal poly-His tagged spermidine synthase expressed in Escherichia coli BL21(DE3) using 50 uM p...More data for this Ligand-Target Pair