Affinity DataIC50: 2.80nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 113nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 285nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 288nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 435nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 445nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 695nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 705nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 775nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 845nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 960nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 1.74E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 2.89E+3nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 5.15E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 5.68E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 9.95E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 1.19E+4nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+4nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+5nMAssay Description:Compound was tested for its ability to displace [3H]-pirenzepine (pir) from M1 Muscarinic receptor in rat cortical tissueMore data for this Ligand-Target Pair