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Found 602 with Last Name = 'gao' and Initial = 'f'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50413477(CHEMBL475226)
Affinity DataKi:  1nMAssay Description:Displacement of [125I](R)-1-(3-iodophenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1Hbenzo[e][1,4]diazepin-3-yl)urea from human CCK2 receptor expresse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193475((3R)-3-{[2-({2-[({[(1S)-1-carbamoyl-4-[(diaminomet...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50292348(CHEMBL501262 | bryostatin 10)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193477(3-((R)-4-(3-(2-(2-(((2R,3S,4R,5R,6R)-5-amino-6-((1...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193484(CID44414951 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193487((3R)-3-[(2-{[2-({[(3-{[3-(dimethylamino)propyl]ami...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193478(CID44415032 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50413478(CHEMBL515288)
Affinity DataKi:  3.72nMAssay Description:Displacement of [125I](S)-1-(3-iodophenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)urea from human CCK1 receptor express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50292349(CHEMBL505767 | bryostatin 18)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193488(CID44415033 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  7.40nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193474((R)-4-(3-(2-(2-(((2R,3S,4R,5R,6R)-5-amino-6-((1R,2...)
Affinity DataKi:  11nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193480((R)-4-(3-(2-(2-(((2R,3S,4R,5R,6R)-5-amino-6-((1R,2...)
Affinity DataKi:  12nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343634(4-((E)-4-((S)-1-((1R,2S,5S)-2-((S)-5-amino-1-(benz...)
Affinity DataKi:  33nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343641(CHEMBL1774964 | cis-4-((E)-4-((S)-4-methyl-1-oxo-1...)
Affinity DataKi:  39nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343632(4-((E)-4-((S)-1-((1R,2S,5S)-2-((S)-5-amino-1-(benz...)
Affinity DataKi:  43nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193476(CID44415023 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  43nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343644(CHEMBL1774967 | cis-4-((E)-4-oxo-4-((S)-1-oxo-1-((...)
Affinity DataKi:  46nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343633(4-((E)-3-((S)-1-((1R,2S,5S)-2-((S)-5-amino-1-(benz...)
Affinity DataKi:  48nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343635(4-((E)-4-((3S,6S)-6-((S)-5-amino-1-(benzylamino)-1...)
Affinity DataKi:  57nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343642(CHEMBL1774965 | cis-4-((E)-4-((S)-1-((1R,2S,5S)-2-...)
Affinity DataKi:  66nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343631(4-((E)-4-((S)-1-((S)-2-((S)-5-amino-1-(benzylamino...)
Affinity DataKi:  66nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193486(CID44415022 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  76nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343639(CHEMBL1774962 | cis-4-((E)-4-((S)-1-((1R,2S,5S)-2-...)
Affinity DataKi:  83nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343638(4-((E)-4-((S)-4-methyl-1-oxo-1-((S)-2-(2-ureidoeth...)
Affinity DataKi:  94nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343645(4-((E)-4-((3S,6S)-6-((R)-5-amino-5-oxopentan-2-ylc...)
Affinity DataKi:  105nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193482(CID44414946 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  110nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343643(CHEMBL1774966 | cis-2-((1R,2S,5S)-3-((S)-2-((E)-3-...)
Affinity DataKi:  114nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50292351(CHEMBL509516 | bryostatin 16)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193479(CID44414949 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  119nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193485((3R)-3-{[2-({2-[({[(5S)-5-acetamido-6-methoxy-6-ox...)
Affinity DataKi:  130nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343636(4-((E)-4-((S)-1-((S)-2-((R)-5-amino-5-oxopentan-2-...)
Affinity DataKi:  144nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193483(CID44415024 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  161nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50413477(CHEMBL475226)
Affinity DataKi:  174nMAssay Description:Displacement of [125I](S)-1-(3-iodophenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)urea from human CCK1 receptor express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343646(2-((3S,6S)-4-oxo-3-((E)-3-(4-(phosphonooxy)phenyl)...)
Affinity DataKi:  188nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50292350(CHEMBL452391 | bryostatin 17 | delta 19,20-bryosta...)
Affinity DataKi:  188nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343640(CHEMBL1774963 | cis-2-((1R,2S,5S)-3-((S)-4-methyl-...)
Affinity DataKi:  193nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343637(2-((S)-1-((S)-4-methyl-2-((E)-3-(4-(phosphonooxy)p...)
Affinity DataKi:  203nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Peking University

Curated by ChEMBL
LigandPNGBDBM50061567(1,1-Dimethyl-4-phenyl-piperazin-1-ium | CHEMBL1347...)
Affinity DataKi:  250nMAssay Description:Binding affinity towards nicotinic receptor in rat brain using [3H]cytisine ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Texas M. D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50343647(4-((E)-4-oxo-4-((3S,6S)-4-oxo-6-(2-ureidoethylcarb...)
Affinity DataKi:  386nMAssay Description:Binding affinity to SH2 domain of Stat3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50413478(CHEMBL515288)
Affinity DataKi:  537nMAssay Description:Displacement of [125I](R)-1-(3-iodophenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1Hbenzo[e][1,4]diazepin-3-yl)urea from human CCK2 receptor expresse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50155579(CHEMBL3546846)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human LSD1 using H3K4Me1 peptide as substrate incubated for 60 min by peroxidase-coupled methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50155579(CHEMBL3546846)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50155579(CHEMBL3546846)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of recombinant human MAO-B using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGNAT family acetyltransferase(Enterococcus durans)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50193481(CID44414945 | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of Enterococcus faecium AAC(6')IiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 2(Homo sapiens (Human))
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50155579(CHEMBL3546846)
Affinity DataKi:  6.10E+4nMAssay Description:Inhibition of human LSD2 using H3K4Me2 peptide as substrate incubated for 60 min by peroxidase-coupled methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM624953(US20230322745, Compound 24)
Affinity DataIC50:  0.0140nMAssay Description:The M2 receptor membrane protein was prepared at 100 μg/mL by Biology Department of WuXi AppTec, and compounds were serially diluted in a 2.5-fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM624955(US20230322745, Compound 25)
Affinity DataIC50:  0.0300nMAssay Description:The M2 receptor membrane protein was prepared at 100 μg/mL by Biology Department of WuXi AppTec, and compounds were serially diluted in a 2.5-fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM624859(US20230322745, Compound 1)
Affinity DataIC50:  0.0620nMAssay Description:The M2 receptor membrane protein was prepared at 100 μg/mL by Biology Department of WuXi AppTec, and compounds were serially diluted in a 2.5-fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM624956(US20230322745, Compound 28)
Affinity DataIC50:  0.0830nMAssay Description:The M2 receptor membrane protein was prepared at 100 μg/mL by Biology Department of WuXi AppTec, and compounds were serially diluted in a 2.5-fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM624948(US20230322745, Compound 15 | US20230322745, Compou...)
Affinity DataIC50:  0.104nMAssay Description:The M2 receptor membrane protein was prepared at 100 μg/mL by Biology Department of WuXi AppTec, and compounds were serially diluted in a 2.5-fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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