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Found 929 with Last Name = 'garlisi' and Initial = 'cg'
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210759(US9290454, 4.4)
Affinity DataKi:  0.230nMAssay Description:Antagonist activity at CRTh2 (unknown origin) assessed as inhibition of CD11b activationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210749(US9290454, 3.1)
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at CRTh2 (unknown origin) assessed as inhibition of CD11b activationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449263(CHEMBL3125333)
Affinity DataKi:  1.10nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210750(US9290454, 3.2)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at CRTh2 (unknown origin) assessed as inhibition of CD11b activationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449259(CHEMBL3125329)
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449257(CHEMBL3125327)
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449258(CHEMBL3125328)
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449277(CHEMBL3125160)
Affinity DataKi:  1.90nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449261(CHEMBL3125331)
Affinity DataKi:  1.90nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449272(CHEMBL3125342)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449278(CHEMBL3125161)
Affinity DataKi:  2.30nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449276(CHEMBL3125159)
Affinity DataKi:  2.5nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449260(CHEMBL3125330)
Affinity DataKi:  2.5nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449255(CHEMBL3125322)
Affinity DataKi:  2.60nMAssay Description:Partial agonist activity at human CRTH2 receptor expressed in HEK cells assessed as forskolin-induced cAMP formation preincubated for 10 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449267(CHEMBL3125337)
Affinity DataKi:  2.60nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449268(CHEMBL3125338)
Affinity DataKi:  3nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449266(CHEMBL3125336)
Affinity DataKi:  3.40nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449264(CHEMBL3125334)
Affinity DataKi:  3.70nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449275(CHEMBL3125158)
Affinity DataKi:  3.70nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449265(CHEMBL3125335)
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449256(CHEMBL3125326)
Affinity DataKi:  4.70nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449283(CHEMBL3125321)
Affinity DataKi:  5.60nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210749(US9290454, 3.1)
Affinity DataKi:  5.80nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210759(US9290454, 4.4)
Affinity DataKi:  5.90nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449270(CHEMBL3125340)
Affinity DataKi:  6nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210750(US9290454, 3.2)
Affinity DataKi:  6.5nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Macaca mulatta)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50161407(CHEMBL178447 | [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-...)
Affinity DataKi:  7.20nMAssay Description:In vitro binding affinity against monkey CC chemokine receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50167438(CHEMBL191464 | Quinoline-6-carboxylic acid [1'-(3,...)
Affinity DataKi:  7.30nMAssay Description:In vitro binding activity against C-C chemokine receptor type 3 using [35S]-GTP-gammaS, as radioligand More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449279(CHEMBL3125162)
Affinity DataKi:  7.40nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449274(CHEMBL3125157)
Affinity DataKi:  7.5nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50161419(CHEMBL178818 | [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-...)
Affinity DataKi:  7.70nMAssay Description:In vitro binding affinity against C-C chemokine receptor type 3 expressing in rat Y3 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50161419(CHEMBL178818 | [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-...)
Affinity DataKi:  7.70nMAssay Description:In vitro binding affinity against C-C chemokine receptor type 3 expressing in rat Y3 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50452163(CHEMBL4208892)
Affinity DataKi:  7.80nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210751(US9290454, 3.3)
Affinity DataKi:  8.5nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210752(US9290454, 3.4)
Affinity DataKi:  9.20nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50452165(CHEMBL4216753)
Affinity DataKi:  11nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449271(CHEMBL3125341)
Affinity DataKi:  11nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50452167(CHEMBL4213820)
Affinity DataKi:  13nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210753(US9290454, 3.5)
Affinity DataKi:  13nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50161415(CHEMBL181460 | [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity against C-C chemokine receptor type 3 expressing in rat Y3 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50161415(CHEMBL181460 | [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity against C-C chemokine receptor type 3 expressing in rat Y3 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210757(US9290454, 4.2)
Affinity DataKi:  14nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449262(CHEMBL3125332)
Affinity DataKi:  14nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210768(US9290454, 8.2)
Affinity DataKi:  15nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50161432(CHEMBL181273 | [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity against C-C chemokine receptor type 3 expressing in rat Y3 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50161420(CHEMBL362040 | [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity against C-C chemokine receptor type 3 expressing in rat Y3 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449281(CHEMBL3125319)
Affinity DataKi:  18nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM210754(US9290454, 3.6 | US9290454, 3.7)
Affinity DataKi:  19nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50161439(CHEMBL181034 | [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-...)
Affinity DataKi:  20nMAssay Description:In vitro binding affinity against C-C chemokine receptor type 3 expressing in rat Y3 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50449282(CHEMBL3125320)
Affinity DataKi:  20nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO-1 cells assessed as inhibition of PGD2-induced Ca2+ flux preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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