Compile Data Set for Download or QSAR
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Found 55 with Last Name = 'geng' and Initial = 'p'
TargetCardiac ryanodine receptor 2(Canis familiaris)
University Of California

Curated by ChEMBL
LigandPNGBDBM50044994(2,6,9,11,13,14-hexahydroxy-11-isopropyl-3,7,10-tri...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity towards ryanodine receptor in canine ventrical preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50051434(10-epi-hydroxy-Ryanodine | CHEMBL308183 | Ryanodin...)
Affinity DataKi:  1.80nMAssay Description:Binding to ryanodine receptor in canine cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50051434(10-epi-hydroxy-Ryanodine | CHEMBL308183 | Ryanodin...)
Affinity DataIC50:  3.30nMAssay Description:Inhibitory activity against ryanodine receptor from mouse brain preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50051434(10-epi-hydroxy-Ryanodine | CHEMBL308183 | Ryanodin...)
Affinity DataIC50:  3.5nMAssay Description:Inhibitory activity against ryanodine receptor from rabbit muscle preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50158869(CHEMBL3786182 | US10836743, Compound GSK-2879552 |...)
Affinity DataIC50:  41nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231781(CHEMBL4090528)
Affinity DataIC50:  564nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231773(CHEMBL4069511)
Affinity DataIC50:  678nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231771(CHEMBL4087193)
Affinity DataIC50:  685nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231780(CHEMBL4065771)
Affinity DataIC50:  717nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231778(CHEMBL4068480)
Affinity DataIC50:  758nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231754(CHEMBL4074390)
Affinity DataIC50:  960nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231769(CHEMBL4094875)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231776(CHEMBL4095820)
Affinity DataIC50:  2.63E+3nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142662(1-Butyl-1-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-di...)
Affinity DataEC50:  7.90nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142669(CHEMBL47953 | [4'-((2S,5S)-1,5-Dimethyl-4-octyl-3,...)
Affinity DataEC50:  1.80nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142680(CHEMBL46216 | N-[4'-((2S,5S)-1,5-Dimethyl-4-octyl-...)
Affinity DataEC50:  9.70nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142682((3R,6R)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142661(CHEMBL47059 | N-Butyl-N-[4'-((2S,5S)-1,5-dimethyl-...)
Affinity DataEC50:  14nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142654(2-{(S)-3-[3'-(1-Butyl-3-methyl-ureidomethyl)-biphe...)
Affinity DataEC50:  1.70nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142672(Butyl-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-dioxo-...)
Affinity DataEC50:  31nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142668((S)-1-Hexyl-4-methyl-3-(3',4',5'-trimethoxy-biphen...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142675(1-Butyl-1-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-di...)
Affinity DataEC50:  7.20nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142660((S)-4-Methyl-1-nonyl-3-(3',4',5'-trimethoxy-biphen...)
Affinity DataEC50:  900nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142663(2-[(S)-2,5-Dioxo-3-(3',4',5'-trimethoxy-biphenyl-4...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142674((3S,6R)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  68nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142664(2-[(S)-2,5-Dioxo-4-propyl-3-(3',4',5'-trimethoxy-b...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142667(2-[(S)-4-Ethyl-2,5-dioxo-3-(3',4',5'-trimethoxy-bi...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142670(1-[4'-((2S,5S)-1,5-Dimethyl-4-octyl-3,6-dioxo-pipe...)
Affinity DataEC50:  3.60nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142676((3S,6S)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  13nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142677((S)-4-Methyl-1-pentyl-3-(3',4',5'-trimethoxy-biphe...)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142671((S)-3-(3',5'-Dimethoxy-biphenyl-4-ylmethyl)-4-meth...)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142666((S)-1-Heptyl-4-methyl-3-(3',4',5'-trimethoxy-biphe...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142679((R)-1-Hexyl-4-methyl-3-(3',4',5'-trimethoxy-biphen...)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142656(Butyl-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-dioxo-...)
Affinity DataEC50:  48nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142676((3S,6S)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  32nMAssay Description:Agonistic activity of the compound was determined in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142675(1-Butyl-1-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-di...)
Affinity DataEC50:  9.5nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142662(1-Butyl-1-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-di...)
Affinity DataEC50:  1.20nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142672(Butyl-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-dioxo-...)
Affinity DataEC50:  2.70nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142657((3S,6S)-1-Heptyl-4,6-dimethyl-3-(3',4',5'-trimetho...)
Affinity DataEC50:  32nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142661(CHEMBL47059 | N-Butyl-N-[4'-((2S,5S)-1,5-dimethyl-...)
Affinity DataEC50:  35nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142656(Butyl-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-dioxo-...)
Affinity DataEC50:  8.90nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142656(Butyl-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-dioxo-...)
Affinity DataEC50:  48nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142681((S)-4-Methyl-1-octyl-3-(3',4',5'-trimethoxy-biphen...)
Affinity DataEC50:  400nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142657((3S,6S)-1-Heptyl-4,6-dimethyl-3-(3',4',5'-trimetho...)
Affinity DataEC50:  25nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142659((S)-3-(3',4'-Dimethoxy-biphenyl-4-ylmethyl)-4-meth...)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142658((S)-3-(4'-Methoxy-3',5'-dimethyl-biphenyl-4-ylmeth...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142665((3S,6S)-1-Hexyl-4,6-dimethyl-3-(3',4',5'-trimethox...)
Affinity DataEC50:  100nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142678(CHEMBL44663 | N-Butyl-N-[4'-((2S,5S)-4-hexyl-1,5-d...)
Affinity DataEC50:  150nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142651(CHEMBL300022 | N-Hexyl-2-[(S)-4-methyl-2,5-dioxo-3...)
Affinity DataEC50:  3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50142673((3R,6S)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  120nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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