Affinity DataKi: 1.80nMAssay Description:Binding affinity towards ryanodine receptor in canine ventrical preparationMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding to ryanodine receptor in canine cardiac membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibitory activity against ryanodine receptor from mouse brain preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibitory activity against ryanodine receptor from rabbit muscle preparationMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 564nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 678nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 685nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 717nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 758nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 960nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)
Curated by ChEMBL
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.90nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 9.70nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 7.20nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 68nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 3.60nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 9.00E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonistic activity of the compound was determined in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.5nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.90nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair