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Found 82 with Last Name = 'gioannini' and Initial = 't'
LigandPNGBDBM50027473(3-Methyl-1-phenethyl-4-(phenyl-propionyl-amino)-pi...)
Affinity DataIC50:  0.25nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
LigandPNGBDBM50021347(CHEMBL12391 | N-(3-Methyl-1-phenethyl-piperidin-4-...)
Affinity DataIC50:  0.600nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224315(CHEMBL2304164)
Affinity DataIC50:  0.600nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021347(CHEMBL12391 | N-(3-Methyl-1-phenethyl-piperidin-4-...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224313(CHEMBL556159)
Affinity DataIC50:  1.40nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataIC50:  1.5nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataIC50:  1.60nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  2nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  2nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225681(CHEMBL611395)
Affinity DataIC50:  2.30nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224315(CHEMBL2304164)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021257(2-[11,15-dimethoxy-3-methyl-(14R)-13-oxa-3-azahexa...)
Affinity DataIC50:  2.5nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225681(CHEMBL611395)
Affinity DataIC50:  3.5nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  4nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  4nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  4.20nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
LigandPNGBDBM50224311(CHEMBL537622)
Affinity DataIC50:  4.40nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224307(CHEMBL539579)
Affinity DataIC50:  5nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224314(CHEMBL174189)
Affinity DataIC50:  5.5nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225690(CHEMBL610808)
Affinity DataIC50:  6nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225684(CHEMBL610611)
Affinity DataIC50:  6nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021255(2-[11,15-dimethoxy-3-methyl-(1R,14R,15R)-13-oxa-3-...)
Affinity DataIC50:  6.40nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225683(CHEMBL610807)
Affinity DataIC50:  7nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225685(CHEMBL175344)
Affinity DataIC50:  8nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224316(CHEMBL171932)
Affinity DataIC50:  8.70nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021258(4-(4-allyloxyphenyl)-2-(11,15-dimethoxy-3-methyl-1...)
Affinity DataIC50:  10nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225692(CHEMBL610612)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225692(CHEMBL610612)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225690(CHEMBL610808)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225683(CHEMBL610807)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  12.5nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  12.5nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  13nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  13nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225682(CHEMBL174530)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224318(CHEMBL535806)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224313(CHEMBL556159)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  27nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
LigandPNGBDBM50225693(CHEMBL369657)
Affinity DataIC50:  30nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  35nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  35nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021257(2-[11,15-dimethoxy-3-methyl-(14R)-13-oxa-3-azahexa...)
Affinity DataIC50:  38nMAssay Description:Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225688(CHEMBL611391)
Affinity DataIC50:  40nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225689(CHEMBL611392)
Affinity DataIC50:  50nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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