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Found 447 with Last Name = 'goettert' and Initial = 'm'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494296(CHEMBL3086685)
Affinity DataIC50:  1nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494284(CHEMBL3087471)
Affinity DataIC50:  1.60nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494256(CHEMBL3087469)
Affinity DataIC50:  1.70nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494261(CHEMBL3087470)
Affinity DataIC50:  1.80nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343492((S)-4-(4-(4-fluorophenyl)-2-(methylsulfinyl)-1H-im...)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343508(4-(4-(4-Fluorophenyl)-2-(methylthio)-1H-imidazol-5...)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343505((S)-4-(4-(4-fluorophenyl)-2-(isopropylsulfinyl)-1H...)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398456(CHEMBL2179119)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398191(CHEMBL2182085)
Affinity DataIC50:  3nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494262(CHEMBL3086686)
Affinity DataIC50:  3nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Eberhard Karls Universit£T T£Bingen

Curated by ChEMBL
LigandPNGBDBM50503009(CHEMBL4526183)
Affinity DataIC50:  3nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Eberhard Karls Universit£T T£Bingen

Curated by ChEMBL
LigandPNGBDBM50503017(CHEMBL4483032)
Affinity DataIC50:  3nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343506((R)-4-(4-(4-fluorophenyl)-2-(isopropylsulfinyl)-1H...)
Affinity DataIC50:  4nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343507(4-(4-(4-Fluorophenyl)-2-(isopropylthio)-1H-imidazo...)
Affinity DataIC50:  4nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398165(CHEMBL2182072)
Affinity DataIC50:  4nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494284(CHEMBL3087471)
Affinity DataIC50:  4nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 300 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50251985(4-(4-(4-fluorophenyl)-2-(methylthio)-1H-imidazol-5...)
Affinity DataIC50:  5nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398153(CHEMBL2177215)
Affinity DataIC50:  5nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343505((S)-4-(4-(4-fluorophenyl)-2-(isopropylsulfinyl)-1H...)
Affinity DataIC50:  6nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50503015(CHEMBL4457174)
Affinity DataIC50:  7nMAssay Description:Inhibition of P38alpha MAPK (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398458(CHEMBL2179117)
Affinity DataIC50:  8nMAssay Description:Inhibition of p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494263(CHEMBL3086680)
Affinity DataIC50:  8nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50330167(2-(4-fluorophenyl)-N-(4-(4-(4-fluorophenyl)-2-(met...)
Affinity DataIC50:  9nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398166(CHEMBL2182071)
Affinity DataIC50:  9nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398187(CHEMBL2182089)
Affinity DataIC50:  10nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398154(CHEMBL2177214)
Affinity DataIC50:  10nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398163(CHEMBL2182074)
Affinity DataIC50:  10nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494273(CHEMBL3087473)
Affinity DataIC50:  10nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343502((R)-4-(4-(4-fluorophenyl)-2-(methylsulfinyl)-1H-im...)
Affinity DataIC50:  11nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343504((R)-N-cyclohexyl-4-(4-(4-fluorophenyl)-2-(isopropy...)
Affinity DataIC50:  11nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398457(CHEMBL2179118)
Affinity DataIC50:  11nMAssay Description:Inhibition of p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398188(CHEMBL2182088)
Affinity DataIC50:  11nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Eberhard Karls Universit£T T£Bingen

Curated by ChEMBL
LigandPNGBDBM50502999(CHEMBL4561980)
Affinity DataIC50:  11nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343489(CHEMBL1773502 | N-Cyclohexyl-4-(4-(4-fluorophenyl)...)
Affinity DataIC50:  12nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343493((R)-4-(4-(4-fluorophenyl)-2-(methylsulfinyl)-1H-im...)
Affinity DataIC50:  12nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50343487((S)-4-(4-(4-fluorophenyl)-2-(methylsulfinyl)-1H-im...)
Affinity DataIC50:  12nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398150(CHEMBL2177106)
Affinity DataIC50:  12nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398186(CHEMBL2182090)
Affinity DataIC50:  12nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398194(CHEMBL2182082)
Affinity DataIC50:  12nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398132(CHEMBL2182099)
Affinity DataIC50:  13nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50392172(CHEMBL2152941)
Affinity DataIC50:  13nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Eberhard Karls Universit£T T£Bingen

Curated by ChEMBL
LigandPNGBDBM50503022(CHEMBL4445449)
Affinity DataIC50:  13nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398151(CHEMBL2177217)
Affinity DataIC50:  14nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398155(CHEMBL2177213)
Affinity DataIC50:  14nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50494258(CHEMBL3086675)
Affinity DataIC50:  14nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of p38 alpha MAPK in human whole blood assessed as phosphorylation of ATF-2 by immunosorbent non-radioactive enzyme assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398464(CHEMBL2179115)
Affinity DataIC50:  15nMAssay Description:Inhibition of p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398173(CHEMBL2177209)
Affinity DataIC50:  15nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50398466(CHEMBL2179128)
Affinity DataIC50:  16nMAssay Description:Inhibition of p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50502996(CHEMBL4451444)
Affinity DataIC50:  16nMAssay Description:Inhibition of P38alpha MAPK (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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