Affinity DataKi: 0.210nM ΔG°: -55.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.220nM ΔG°: -55.1kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.370nM ΔG°: -53.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [125I]-apelin-13 from human APJ receptor stably expressed in CHOK1 cell membrane measured after 2 hrs by topcount scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 1.15nM ΔG°: -51.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.62nM ΔG°: -50.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 1.66nM ΔG°: -50.1kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.29nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 2.57nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nM ΔG°: -48.9kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 2.88nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.31nM ΔG°: -48.4kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.37nM ΔG°: -47.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.76nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.76nM ΔG°: -46.3kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.91nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11.2nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 12nM ΔG°: -45.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair