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Found 250 with Last Name = 'gopalakrishnan' and Initial = 'r'
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM36609(Rapamycin C-7, analog 4 | SIROLIMUS | US11603377, ...)
Affinity DataKi:  3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432752(FK-506)
Affinity DataKi:  80nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388298(CHEMBL2058794)
Affinity DataKi:  200nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432732(CHEMBL2348594)
Affinity DataKi:  300nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432739(CHEMBL2348604)
Affinity DataKi:  500nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432736(CHEMBL2348607)
Affinity DataKi:  870nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432740(CHEMBL2348599)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432748(CHEMBL2348587)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432735(CHEMBL2348608)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432745(CHEMBL2348591)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50132556((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432738(CHEMBL2348605)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432734(CHEMBL2348592)
Affinity DataKi:  7.60E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432747(CHEMBL2348588)
Affinity DataKi:  8.80E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432742(CHEMBL2348597)
Affinity DataKi:  9.80E+3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388280(CHEMBL2058234)
Affinity DataKi:  1.38E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432733(CHEMBL2348593)
Affinity DataKi:  1.39E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432739(CHEMBL2348604)
Affinity DataKi:  1.81E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432749(CHEMBL2348611)
Affinity DataKi:  2.37E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432743(CHEMBL2348596)
Affinity DataKi:  2.70E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432737(CHEMBL2348606)
Affinity DataKi:  2.77E+4nMAssay Description:Binding affinity to FKBP12 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432750(CHEMBL2348610)
Affinity DataKi:  5.11E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432746(CHEMBL2348590)
Affinity DataKi:  6.48E+4nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432741(CHEMBL2348598)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432738(CHEMBL2348605)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432737(CHEMBL2348606)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432735(CHEMBL2348608)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432751(CHEMBL2348609)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388294(CHEMBL2058790)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432744(CHEMBL2348595)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388295(CHEMBL2058791)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50432736(CHEMBL2348607)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388300(CHEMBL2058796)
Affinity DataIC50:  3nMAssay Description:Binding affinity to FKBP12 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50109811((S)-1-[2-Oxo-2-(3,4,5-trimethoxy-phenyl)-acetyl]-p...)
Affinity DataIC50:  17nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388293(CHEMBL2058787)
Affinity DataIC50:  21nMAssay Description:Binding affinity to FKBP12 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388324(CHEMBL2059238)
Affinity DataIC50:  50nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388325(CHEMBL2059239)
Affinity DataIC50:  60nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388323(CHEMBL2059237)
Affinity DataIC50:  60nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388314(CHEMBL2059029)
Affinity DataIC50:  60nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388318(CHEMBL2057227)
Affinity DataIC50:  60nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388314(CHEMBL2059029)
Affinity DataIC50:  60nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388323(CHEMBL2059237)
Affinity DataIC50:  60nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388311(CHEMBL2059026)
Affinity DataIC50:  100nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388309(CHEMBL2059024)
Affinity DataIC50:  100nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50132556((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataIC50:  114nMAssay Description:Binding affinity to FKBP12 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388298(CHEMBL2058794)
Affinity DataIC50:  115nMAssay Description:Binding affinity to FKBP12 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388312(CHEMBL2059027)
Affinity DataIC50:  150nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50132556((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataIC50:  170nMAssay Description:Binding affinity to FKBP12 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388295(CHEMBL2058791)
Affinity DataIC50:  200nMAssay Description:Binding affinity to FKBP12 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50388289(CHEMBL2058495)
Affinity DataIC50:  230nMAssay Description:Binding affinity to FKBP12 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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