Affinity DataKi: 0.400nMAssay Description:Binding affinity to human recombinant GnRH receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to rat pituitary GnRH receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 4.20nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Competitive inhibition of GnRH-stimulated extracellular acidification in cells expressing recombinant rat GnRH receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 5.40nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 5.90nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 6.5nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 7.70nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 7.90nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 9.5nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 10nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 10nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 12nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 13nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 18nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 45nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Isomerase Therapeutics
US Patent
Isomerase Therapeutics
US Patent
Affinity DataKi: 95nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair