Affinity DataKi: 0.200nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 13.4nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair