Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.360nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Leukotriene D4 induced contraction of guinea-pig trachea was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration of the compound against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined (Experiment 2)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at human CRF1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration of the compound against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined (Experiment 1)More data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor-binding protein(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity to CRF-binding protein (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Sage Therapeutics
Curated by ChEMBL
Sage Therapeutics
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Kv1.5 (unknown origin) by patch clamp assayMore data for this Ligand-Target Pair