TargetDihydrofolate reductase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari
Curated by ChEMBL
Universita` Degli Studi Di Sassari
Curated by ChEMBL
Affinity DataKi: 0.000340nMAssay Description:Inhibition of human DHFR by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
The M. S. University Of Baroda
Curated by ChEMBL
The M. S. University Of Baroda
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity to amyloid beta (1 to 40) (unknown origin) aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda
Curated by ChEMBL
The M. S. University Of Baroda
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
The M. S. University Of Baroda
Curated by ChEMBL
The M. S. University Of Baroda
Curated by ChEMBL
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Binding affinity to amyloid beta (1 to 40) (unknown origin) fibrilsMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
The M. S. University Of Baroda
Curated by ChEMBL
The M. S. University Of Baroda
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Ki value for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Ki value for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 6.91nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 6.97nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Banaras Hindu University
Curated by ChEMBL
Banaras Hindu University
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 30 mins followed by substrate addition b...More data for this Ligand-Target Pair
Affinity DataKi: 7.07nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 12.3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 12.4nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) measured by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:A solution of the L-FABP (500 nM) and ANS (35 µM) was titrated with phytanic acid (0-6.4 µM) or fenofibrate (0-6 µM for the rat L-FABP...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:A solution of the L-FABP (500 nM) and ANS (35 µM) was titrated with phytanic acid (0-6.4 µM) or fenofibrate (0-6 µM for the rat L-FABP...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to amyloid beta (1 to 40) (unknown origin) fibrilsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
The M. S. University Of Baroda
Curated by ChEMBL
The M. S. University Of Baroda
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Competitive inhibition of human MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH as substrate preincubated for 60 mins followed by substrate addition by...More data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
TargetRibonuclease pancreatic(Bison bison (American bison))
Indian Institute Of Technology
Curated by ChEMBL
Indian Institute Of Technology
Curated by ChEMBL
Affinity DataKi: 27nMpH: 5.9Assay Description:Inhibition of bovine pancreatic RNase A at pH 5.9 by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 31.3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 31.7nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:A solution of the L-FABP (500 nM) and ANS (35 µM) was titrated with phytanic acid (0-6.4 µM) or fenofibrate (0-6 µM for the rat L-FABP...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Indian Institute Of Technology (Bhu)
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Binding affinity to amyloid beta (1 to 42) (unknown origin) aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:A solution of the L-FABP (500 nM) and ANS (35 µM) was titrated with phytanic acid (0-6.4 µM) or fenofibrate (0-6 µM for the rat L-FABP...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:A solution of the L-FABP (500 nM) and ANS (35 µM) was titrated with phytanic acid (0-6.4 µM) or fenofibrate (0-6 µM for the rat L-FABP...More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M2 receptor in rat heartMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetRibonuclease pancreatic(Bison bison (American bison))
Indian Institute Of Technology
Curated by ChEMBL
Indian Institute Of Technology
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Inhibition of bovine pancreatic RNase A by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M3 receptor in rat submandibular glandMore data for this Ligand-Target Pair