Compile Data Set for Download or QSAR
maximum 50k data
Found 565 with Last Name = 'haudecoeur' and Initial = 'r'
LigandPNGBDBM50608949(CHEMBL5270056)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608952(CHEMBL5279881)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608953(CHEMBL5284094)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608950(CHEMBL5280131)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608951(CHEMBL5277645)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608941(CHEMBL5280240)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50407853(CHEMBL94644)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM85862(1-(2-Chloro-3,4-dimethoxybenzyl)-6-methyl-2,3,4,9-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50407849(CHEMBL96480)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608955(CHEMBL96427)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608956(CHEMBL94655)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608954(CHEMBL329479)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50007554(4-Methoxymethyl-6-propoxy-9H-beta-carboline-3-carb...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608939(CHEMBL5266498)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50007554(4-Methoxymethyl-6-propoxy-9H-beta-carboline-3-carb...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha2 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50000177(7,12-Dihydro-5,7,12-triaza-indeno[1,2-a]fluorene |...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha3 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50000177(7,12-Dihydro-5,7,12-triaza-indeno[1,2-a]fluorene |...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608941(CHEMBL5280240)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha2 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608942(CHEMBL5290579)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha5 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50329657(6-Ethynl-9H-beta-carboline-3-carboxylic acid t-but...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataKi:  1nMAssay Description:Binding affinity to MAO-A (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
LigandPNGBDBM50244035(Beta CCE | CHEMBL454606 | cid_105078 | ethyl 9H-py...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50000177(7,12-Dihydro-5,7,12-triaza-indeno[1,2-a]fluorene |...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha2 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50244033(Abecarnil | CHEMBL454095 | isopropyl 6-(benzyloxy)...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50007554(4-Methoxymethyl-6-propoxy-9H-beta-carboline-3-carb...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human recombinant GABAA alpha5 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50007554(4-Methoxymethyl-6-propoxy-9H-beta-carboline-3-carb...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human recombinant GABAA alpha3 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50244033(Abecarnil | CHEMBL454095 | isopropyl 6-(benzyloxy)...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human recombinant GABAA alpha2 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608941(CHEMBL5280240)
Affinity DataKi:  2nMAssay Description:Binding affinity to human recombinant GABAA alpha3 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608940(CHEMBL5290464)
Affinity DataKi:  2nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608936(CHEMBL510764)
Affinity DataKi:  2nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50243981(Beta CCM | CHEMBL453066 | Methyl Beta-carboline-3 ...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608946(CHEMBL2008708)
Affinity DataKi:  2nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608945(CHEMBL497197)
Affinity DataKi:  3nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50407849(CHEMBL96480)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2C expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608943(CHEMBL5275690)
Affinity DataKi:  3nMAssay Description:Binding affinity to human recombinant GABAA alpha5 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608947(CHEMBL5281056)
Affinity DataKi:  3nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608939(CHEMBL5266498)
Affinity DataKi:  3nMAssay Description:Binding affinity to human recombinant GABAA alpha2 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM85039(CAS_121926 | NSC_121926 | ZK 93423)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50244033(Abecarnil | CHEMBL454095 | isopropyl 6-(benzyloxy)...)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant GABAA alpha3 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608944(CHEMBL496990)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM85039(CAS_121926 | NSC_121926 | ZK 93423)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant GABAA alpha2 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50125136(2-[2,3']Bipyridinyl-6'-yl-1-(2,3-dihydro-benzofura...)
Affinity DataKi:  4nMAssay Description:Binding affinity to PDE5 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608942(CHEMBL5290579)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant GABAA alpha3 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608941(CHEMBL5280240)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant GABAA alpha5 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608943(CHEMBL5275690)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant GABAA alpha3 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608938(CHEMBL5290746)
Affinity DataKi:  5nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50608937(CHEMBL2262044)
Affinity DataKi:  5nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50244033(Abecarnil | CHEMBL454095 | isopropyl 6-(benzyloxy)...)
Affinity DataKi:  5nMAssay Description:Binding affinity to human recombinant GABAA alpha5 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50608939(CHEMBL5266498)
Affinity DataKi:  5nMAssay Description:Binding affinity to human recombinant GABAA alpha3 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Displayed 1 to 50 (of 565 total ) | Next | Last >>
Jump to: