BindingDB PrimarySearch_ki

Found 1266 with Last Name = 'heering' and Initial = 'j'

Leukotriene A-4 hydrolase(Homo sapiens (Human))
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50116538(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-pro...)

Ki: 3nMAssay Description:Non-competitive inhibition of human C-terminal his6-tagged/N-terminal T7 gene leader sequence-tagged LTA4H using varying levels of L-arginine-7-amino...More data for this Ligand-Target Pair

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3D Structure (crystal)

Leukotriene A-4 hydrolase(Homo sapiens (Human))
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50197085(CHEMBL3921982)

Ki: 160nMAssay Description:Competitive inhibition of human C-terminal his6-tagged/N-terminal T7 gene leader sequence-tagged LTA4H using varying levels of L-arginine-7-amino-4-M...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Leukotriene A-4 hydrolase(Homo sapiens (Human))
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)

Ki: 320nMAssay Description:Competitive inhibition of human C-terminal his6-tagged/N-terminal T7 gene leader sequence-tagged LTA4H using varying levels of L-arginine-7-amino-4-M...More data for this Ligand-Target Pair

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3D Structure (crystal)

Leukotriene A-4 hydrolase(Homo sapiens (Human))
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50197084(CHEMBL3883608)

Ki: 360nMAssay Description:Competitive inhibition of human C-terminal his6-tagged/N-terminal T7 gene leader sequence-tagged LTA4H using varying levels of L-arginine-7-amino-4-M...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575781(CHEMBL4851364)

Ki: 3.30E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Leukotriene A-4 hydrolase(Homo sapiens (Human))
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)

Ki: 3.70E+3nMAssay Description:Competitive inhibition of human C-terminal his6-tagged/N-terminal T7 gene leader sequence-tagged LTA4H using varying levels of L-arginine-7-amino-4-M...More data for this Ligand-Target Pair

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PDB

3D Structure (crystal)

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575831(CHEMBL4852281)

Ki: 4.20E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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Details Article PubMed

Bifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50530480(CHEMBL4445524)

Ki: 4.80E+3nMAssay Description:Competitive inhibition of full length human soluble epoxide hydrolase pre-incubated for 30 mins before DiFMUP substrate addition by fluorescence base...More data for this Ligand-Target Pair

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Bifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50530480(CHEMBL4445524)

Ki: 4.80E+3nMAssay Description:Competitive inhibition of full length human soluble epoxide hydrolase pre-incubated for 30 mins before DiFMUP substrate addition by fluorescence base...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575831(CHEMBL4852281)

Ki: 6.40E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575821(CHEMBL4861964)

Ki: 7.20E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575825(CHEMBL4878621)

Ki: 7.40E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575825(CHEMBL4878621)

Ki: 7.50E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575781(CHEMBL4851364)

Ki: 8.10E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575818(CHEMBL4878719)

Ki: 8.80E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50226181((3R,4S,5R,6R)-5-hydroxy-6-(4-hydroxy-3-(4-hydroxy-...)

Ki: 8.80E+3nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575829(CHEMBL4856665)

Ki: 1.00E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575830(CHEMBL4854132)

Ki: 1.09E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575787(CHEMBL4865071)

Ki: 1.20E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575788(CHEMBL4856823)

Ki: 1.20E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575829(CHEMBL4856665)

Ki: 1.23E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575796(CHEMBL4860932)

Ki: 1.30E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575789(CHEMBL4875925)

Ki: 1.30E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575813(CHEMBL4869659)

Ki: 1.32E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575785(CHEMBL4851932)

Ki: 1.33E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575826(CHEMBL4859492)

Ki: 1.34E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575828(CHEMBL4875883)

Ki: 1.38E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575788(CHEMBL4856823)

Ki: 1.40E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575787(CHEMBL4865071)

Ki: 1.40E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575821(CHEMBL4861964)

Ki: 1.48E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575826(CHEMBL4859492)

Ki: 1.50E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575830(CHEMBL4854132)

Ki: 1.56E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575785(CHEMBL4851932)

Ki: 1.57E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575813(CHEMBL4869659)

Ki: 1.60E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575820(CHEMBL4873678)

Ki: 1.67E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575796(CHEMBL4860932)

Ki: 1.70E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575789(CHEMBL4875925)

Ki: 1.70E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575828(CHEMBL4875883)

Ki: 1.76E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575809(CHEMBL4847717)

Ki: 1.80E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575795(CHEMBL4876524)

Ki: 1.80E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575820(CHEMBL4873678)

Ki: 1.89E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575812(CHEMBL4853160)

Ki: 1.93E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50226181((3R,4S,5R,6R)-5-hydroxy-6-(4-hydroxy-3-(4-hydroxy-...)

Ki: 1.93E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575827(CHEMBL4864565)

Ki: 1.97E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575809(CHEMBL4847717)

Ki: 2.00E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575786(CHEMBL4877664)

Ki: 2.00E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575790(CHEMBL4867942)

Ki: 2.00E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575812(CHEMBL4853160)

Ki: 2.18E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3A(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575827(CHEMBL4864565)

Ki: 2.26E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3A by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Microtubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL

PNG

BDBM50575795(CHEMBL4876524)

Ki: 2.30E+4nMAssay Description:Displacement of sGFP-p62-LIR peptide from human N-terminal SNAP-fused LC3B by time-resolved FRET assayMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Displayed 1 to 50 (of 1266 total ) | Next | Last >>

Filter my 1266 hits

Targets 27▿
- Bifunctional epoxide hydrolase 2 228
- Peroxisome proliferator-activated receptor gamma 207
- Bile acid receptor 91
- Retinoic acid receptor RXR-alpha 90
- Microtubule-associated proteins 1A/1B light chain 3A 90
- Microtubule-associated proteins 1A/1B light chain 3B 82
- Peroxisome proliferator-activated receptor alpha 72
- Retinoic acid receptor RXR-beta 66
- Retinoic acid receptor RXR-gamma 60
- Leukotriene B4 receptor 2 53
- Nuclear receptor subfamily 4 group A member 2 51
- Peroxisome proliferator-activated receptor delta 41
- Polyunsaturated fatty acid 5-lipoxygenase 35
- Nuclear receptor subfamily 2 group E member 1 30
- Leukotriene A-4 hydrolase 25
- Type-1 angiotensin II receptor 12
- Thyroid hormone receptor alpha 6
- Prostaglandin G/H synthase 2 4
- Prostaglandin G/H synthase 1 4
- Thyroid hormone receptor beta 4
- Prothrombin 3
- Retinoic acid receptor alpha 2
- Oxysterols receptor LXR-beta 2
- Oxysterols receptor LXR-alpha 2
- Nuclear receptor subfamily 1 group I member 3 2
- Retinoic acid receptor gamma 2
- Retinoic acid receptor beta 2
- ...
Publications 21▿
- J Med Chem 62: 2112-2126 (2019) 256
- J Med Chem 64: 3720-3746 (2021) 172
- J Med Chem 64: 17259-17276 (2021) 105
- ACS Med Chem Lett 10: 203-208 (2019) 87
- J Med Chem 60: 7703-7724 (2017) 81
- J Med Chem 63: 11498-11521 (2020) 79
- J Med Chem 59: 61-81 (2016) 77
- J Med Chem 62: 8443-8460 (2019) 54
- J Med Chem 63: 4555-4561 (2020) 52
- J Med Chem 60: 7199-7205 (2017) 48
- J Med Chem 63: 11548-11572 (2020) 41
- J Med Chem 64: 15126-15140 (2021) 35
- J Med Chem 63: 6727-6740 (2020) 32
- Bioorg Med Chem 27: (2019) 28
- Bioorg Med Chem 24: 5243-5248 (2016) 25
- ACS Med Chem Lett 12: 1261-1266 (2021) 24
- J Med Chem 64: 8727-8738 (2021) 18
- J Med Chem 64: 2659-2668 (2021) 16
- J Med Chem 63: 10908-10920 (2020) 15
- J Med Chem 65: 2288-2296 (2022) 12
- J Med Chem 64: 2815-2828 (2021) 9
Institutions 9▿
- Goethe-University Frankfurt 646
- Goethe University Frankfurt 303
- Goethe-University 105
- Goethe-University Of Frankfurt 79
- Fraunhofer Ime 41
- Fraunhofer Institute For Molecular Biology And Applied Ecology Ime 28
- Goethe University 25
- Fraunhofer Institute For Translational Medicine And Phamacology Itmp 24
- New York University 15
Affinity: 0.30 to 9.2E+5 nM▿
- Ki 111
- IC50 405
- Kd 59
- EC50 691
- Affinity ≤ nM
Xtal structures: 28
Docked structures: 4
Catalog Cmpds: 102