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Found 630 with Last Name = 'hey' and Initial = 'ja'
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325449(1-(2-(piperidin-1-yl)ethyl)-3-(1-(1-(pyridin-4-ylm...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175828(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325450(1-(2-(dimethylamino)ethyl)-3-(1-(1-(pyridin-4-ylme...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325465(1-benzyl-3-(1-(1-(pyridin-4-ylmethyl)piperidine-4-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325466(1-(3-(dimethylamino)propyl)-3-(1-(1-(pyridin-4-ylm...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175843(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116083(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325460(1-(4-methoxybenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pi...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116091(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116074(CHEMBL66635 | N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325461(1-(3-methoxybenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pi...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116082(3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116076(CHEMBL441252 | N-[5-(3-Carbamoylmethyl-2-oxo-[1,4'...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50116078(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50116078(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116080(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116078(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116074(CHEMBL66635 | N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325473(1-isobutyl-3-(1-(1-(pyridin-4-ylmethyl)piperidine-...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175833(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175843(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM22542(4-(1H-imidazol-4-ylmethyl)piperidine | 4-(1H-imida...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50123075(4-Fluoro-2-{5-[4-(5-fluoro-1H-indol-3-yl)-3,6-dihy...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50103826(7-[4-(6-Hydroxy-biphenyl-3-ylmethyl)-piperazin-1-y...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50020174(1-Benzofuran-7-yl-4-[5-(4-fluoro-phenyl)-1H-pyrrol...)
Affinity DataKi:  0.420nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50020174(1-Benzofuran-7-yl-4-[5-(4-fluoro-phenyl)-1H-pyrrol...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50103839(7-{4-[4-(4-Fluoro-phenyl)-pyridin-2-ylmethyl]-pipe...)
Affinity DataKi:  0.470nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441652(CHEMBL2437433)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325448(1-(2-morpholinoethyl)-3-(1-(1-(pyridin-4-ylmethyl)...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116090(1-(2-{1'-[5-[(3,5-Dichloro-benzoyl)-ethyl-amino]-3...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116088(3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116082(3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50123069(2-(4-(4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridi...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441649(CHEMBL2437416)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325469(1-(2-isopropoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50020177(1-(3,4-Dihydro-2H-benzo[b][1,4]dioxepin-6-yl)-4-(5...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116080(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.700nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441646(CHEMBL2437421)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116090(1-(2-{1'-[5-[(3,5-Dichloro-benzoyl)-ethyl-amino]-3...)
Affinity DataKi:  0.700nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50020182(1-(2-Methoxy-phenyl)-4-(5-phenyl-1H-pyrrol-2-ylmet...)
Affinity DataKi:  0.760nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116091(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116087(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116087(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116076(CHEMBL441252 | N-[5-(3-Carbamoylmethyl-2-oxo-[1,4'...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116075(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325467(1-(3-ethoxypropyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50123081(4-Fluoro-2-{5-[4-(1H-indol-3-yl)-3,6-dihydro-2H-py...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116075(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116083(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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