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Found 10 with Last Name = 'hisaka' and Initial = 'a'
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390982(CHEMBL2075008)
Affinity DataKi:  1.01E+3nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390985(CHEMBL2074707)
Affinity DataKi:  8.32E+3nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390987(CHEMBL2074660)
Affinity DataKi:  4.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390983(CHEMBL2074699)
Affinity DataKi:  5.41E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390984(CHEMBL2074702)
Affinity DataKi:  6.55E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataKi:  8.41E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-485 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390986(CHEMBL2074710)
Affinity DataKi:  8.54E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSqualene synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285068((S)-2-{[(1S,2S)-3-(3,4-Dichloro-phenyl)-2-(2-fluor...)
Affinity DataIC50:  0.520nMAssay Description:Inhibitory activity of the compound against squalene synthase (SQS) obtained from HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSqualene synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288819((R)-4-[(E)-(1S,2S)-2-(3,4-Dichloro-benzyl)-1-methy...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory activity of the compound against squalene synthase (SQS) obtained from HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSqualene synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288818((R)-4-[(1S,2S)-3-(3,4-Dichloro-phenyl)-2-(2-fluoro...)
Affinity DataIC50:  3.90nMAssay Description:Inhibitory activity of the compound against squalene synthase (SQS) obtained from HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails Article