Affinity DataKi: 10nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 93.3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 174nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 309nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 427nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 617nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 676nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 676nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 851nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 891nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 891nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.09E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.34E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.31E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.01E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.37E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant AurKA after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Inhibition of human recombinant AurKB after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of Antwerp
Curated by ChEMBL
University of Antwerp
Curated by ChEMBL
Affinity DataIC50: 167nMAssay Description:Inhibition of human recombinant RIPK1 after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of Antwerp
Curated by ChEMBL
University of Antwerp
Curated by ChEMBL
Affinity DataIC50: 178nMAssay Description:Inhibition of human recombinant RIPK1 after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of Antwerp
Curated by ChEMBL
University of Antwerp
Curated by ChEMBL
Affinity DataIC50: 208nMAssay Description:Inhibition of RIPK1 in mouse L929sA cells transfected with human Fas assessed as inhibition in TNF-induced necroptosis pretreated for 24 hrs followed...More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant AurKA after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 229nMAssay Description:Inhibition of human recombinant AurKB after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 293nMAssay Description:Inhibition of human recombinant AurKA after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of Antwerp
Curated by ChEMBL
University of Antwerp
Curated by ChEMBL
Affinity DataIC50: 295nMAssay Description:Inhibition of human recombinant RIPK1 after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of human recombinant AurKA after 4 hrs by ADP-Glo assayMore data for this Ligand-Target Pair