TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity for phenylethanolamine N-methyl-transferase was determined.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against alpha-2-adrenergic receptor using 10 nM [3H]yohimbine in human platelet membranes from three separate experiments using 10 i...More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Binding affinity against alpha-2-adrenergic receptor using 10 nM [3H]yohimbine in human platelet membranes from three separate experiments using 10 i...More data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity for phenylethanolamine N-methyl-transferase was determined.More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity against alpha-2-adrenergic receptor using 10 nM [3H]yohimbine in human platelet membranes from three separate experiments using 10 i...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibitory activity against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibitory activity against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity against alpha-2-adrenergic receptor using 10 nM [3H]yohimbine in human platelet membranes from four to five separate experiments usi...More data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Inhibitory activity against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 232nMAssay Description:Binding affinity against alpha-2-adrenergic receptor using 10 nM [3H]yohimbine in preparations in human platelet membranes from three separate experi...More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibitory activity against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 338nMAssay Description:Binding affinity against alpha-2-adrenergic receptor using 10 nM [3H]yohimbine in human platelet membranes from three separate experiments using 10 i...More data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.53E+3nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory concentration against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibitory concentration against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
TargetAdenylate cyclase type 1/Adenylate cyclase type 2/Adenylate cyclase type 3/Adenylate cyclase type 4/Adenylate cyclase type 5/Adenylate cyclase type 6/Adenylate cyclase type 8/Adenylyl cyclase 7(Rattus norvegicus)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory concentration against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibitory concentration against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of p60v-abl tyrosine kinase from Abelson murine leukemia virusMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of p60v-abl tyrosine kinase from Abelson murine leukemia virusMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of p60v-abl tyrosine kinase from Abelson murine leukemia virusMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of p60v-abl tyrosine kinase from Abelson murine leukemia virusMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of p60v-abl tyrosine kinase from Abelson murine leukemia virusMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of p60v-abl tyrosine kinase from Abelson murine leukemia virusMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of p60v-abl tyrosine kinase from Abelson murine leukemia virusMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of p60v-abl tyrosine kinase from Abelson murine leukemia virusMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase transforming protein Abl(Abelson murine leukemia virus)
Smith Kline & French Laboratories
Curated by ChEMBL
Smith Kline & French Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of p60-vabl tyrosine kinase isolated from Abelson murine leukemia virus (A-MuLV)More data for this Ligand-Target Pair
Affinity DataEC50: 6.5nMAssay Description:Agonist activity at human kappa opioid receptor-Galpha16 fusion protein expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.810nMAssay Description:Agonist activity at human kappa opioid receptor-Galpha16 fusion protein expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells by [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 385nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells by [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 3.34nMAssay Description:Agonist activity at human kappa opioid receptor assessed as inhibition of Galpha16-induced calcium fluxMore data for this Ligand-Target Pair