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Found 76 with Last Name = 'holloway' and Initial = 'ac'
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509915(CHEMBL4441579)
Affinity DataKi:  8nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50023460(CHEMBL3326517)
Affinity DataKi:  20nMAssay Description:Reversible inhibition of recombinant human CYP19A1 assessed as inhibition of DBF conversion to fluorescein by-product by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442766(CHEMBL2443358)
Affinity DataKi:  20nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442776(CHEMBL2443348)
Affinity DataKi:  20nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50023460(CHEMBL3326517)
Affinity DataKi:  22nMAssay Description:Reversible inhibition of recombinant human CYP19A1 assessed as inhibition of DBF conversion to fluorescein by-product by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509909(CHEMBL4450923)
Affinity DataKi:  24nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50314498(CHEMBL1089299 | N-((2S,3S)-2-(benzo[d][1,3]dioxol-...)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant CYP3A4 assessed as biotransformation of 7-hydroxyquinoline to 7-benzyloxyquinoline measured every minute for 15 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50023465(CHEMBL3326520)
Affinity DataKi:  30nMAssay Description:Inhibition of recombinant human CYP19A1 assessed as inhibition of DBF conversion to fluorescein by-product by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50300539(CHEMBL573430 | N-((2R,3R)-2-(benzo[d][1,3]dioxol-5...)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant CYP3A4 assessed as biotransformation of 7-benzyloxyquinoline to 7-hydroxyquinoline measured every 15 mins by fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50023465(CHEMBL3326520)
Affinity DataKi:  30nMAssay Description:Inhibition of recombinant human CYP19A1 assessed as inhibition of DBF conversion to fluorescein by-product by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509907(CHEMBL4545917)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50360383(CHEMBL1933700)
Affinity DataKi:  50nMAssay Description:Inhibition of human recombinant aromatase assessed as conversion of O-dibenzylfluorescein benzyl ester substrate to fluorescein byproduct by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509911(CHEMBL4561656)
Affinity DataKi:  57nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50360381(CHEMBL1933694)
Affinity DataKi:  60nMAssay Description:Inhibition of human recombinant aromatase assessed as conversion of O-dibenzylfluorescein benzyl ester substrate to fluorescein byproduct by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50314501(((4S,5S)-5-((1S,2S)-3-benzamido-2-(benzo[d][1,3]di...)
Affinity DataKi:  70nMAssay Description:Inhibition of human recombinant CYP3A4 assessed as biotransformation of 7-hydroxyquinoline to 7-benzyloxyquinoline measured every minute for 15 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50300543(((4S,5S)-5-((1R,2R)-3-benzamido-2-(benzo[d][1,3]di...)
Affinity DataKi:  70nMAssay Description:Inhibition of human recombinant CYP3A4 assessed as biotransformation of 7-benzyloxyquinoline to 7-hydroxyquinoline measured every 15 mins by fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442767(CHEMBL2443357)
Affinity DataKi:  70nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509910(CHEMBL4468933)
Affinity DataKi:  74nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509914(CHEMBL4526477)
Affinity DataKi:  79nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50360382(CHEMBL1933699)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant aromatase assessed as conversion of O-dibenzylfluorescein benzyl ester substrate to fluorescein byproduct by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442777(CHEMBL2443365)
Affinity DataKi:  80nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509916(CHEMBL4468397)
Affinity DataKi:  81nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442770(CHEMBL2443354)
Affinity DataKi:  90nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509918(CHEMBL4453517)
Affinity DataKi:  97nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50360380(CHEMBL1933693)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant aromatase assessed as conversion of O-dibenzylfluorescein benzyl ester substrate to fluorescein byproduct by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509913(CHEMBL4437348)
Affinity DataKi:  100nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442771(CHEMBL2443353)
Affinity DataKi:  110nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442775(CHEMBL2443349)
Affinity DataKi:  111nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509912(CHEMBL4562457)
Affinity DataKi:  125nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442764(CHEMBL2443360)
Affinity DataKi:  130nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50023463(CHEMBL3326522)
Affinity DataKi:  145nMAssay Description:Inhibition of recombinant human CYP19A1 assessed as inhibition of DBF conversion to fluorescein by-product by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50023463(CHEMBL3326522)
Affinity DataKi:  150nMAssay Description:Inhibition of recombinant human CYP19A1 assessed as inhibition of DBF conversion to fluorescein by-product by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442768(CHEMBL2443356)
Affinity DataKi:  160nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50300538(CHEMBL574914 | N-((2R,3R)-2-(benzo[d][1,3]dioxol-5...)
Affinity DataKi:  170nMAssay Description:Inhibition of human recombinant CYP3A4 assessed as biotransformation of 7-benzyloxyquinoline to 7-hydroxyquinoline measured every 15 mins by fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442773(CHEMBL2443351)
Affinity DataKi:  170nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509917(CHEMBL4454530)
Affinity DataKi:  180nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442765(CHEMBL2443359)
Affinity DataKi:  200nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50293601((1S,2S,3a1S,12bS)-2-(tert-butyldimethylsilyloxy)-2...)
Affinity DataKi:  210nMAssay Description:Inhibition of human CYP3A4 assessed as biotransformation of 7-benzyloxyquinolineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442769(CHEMBL2443355)
Affinity DataKi:  237nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50314499(CHEMBL1089300 | tert-butyl(2S,3S)-2-(benzo[d][1,3]...)
Affinity DataKi:  240nMAssay Description:Inhibition of human recombinant CYP3A4 assessed as biotransformation of 7-hydroxyquinoline to 7-benzyloxyquinoline measured every minute for 15 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50360384(CHEMBL1933701)
Affinity DataKi:  250nMAssay Description:Inhibition of human recombinant aromatase assessed as conversion of O-dibenzylfluorescein benzyl ester substrate to fluorescein byproduct by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50293600((1S,2S,3a1S,12bS)-2-(tert-butyldimethylsilyloxy)-2...)
Affinity DataKi:  260nMAssay Description:Inhibition of human CYP3A4 assessed as biotransformation of 7-benzyloxyquinolineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50509908(CHEMBL4582591)
Affinity DataKi:  290nMAssay Description:Inhibition of recombinant human CYP19A1 using DBF as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50300541(CHEMBL583953 | tert-butyl(2R,3R)-2-(benzo[d][1,3]d...)
Affinity DataKi:  320nMAssay Description:Inhibition of human recombinant CYP3A4 assessed as biotransformation of 7-benzyloxyquinoline to 7-hydroxyquinoline measured every 15 mins by fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442774(CHEMBL2443350)
Affinity DataKi:  330nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50442762(CHEMBL2443362)
Affinity DataKi:  350nMAssay Description:Inhibition of recombinant human aromatase using O-dibenzylfluorescein benzyl ester as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50023464(CHEMBL3326521)
Affinity DataKi:  355nMAssay Description:Inhibition of recombinant human CYP19A1 assessed as inhibition of DBF conversion to fluorescein by-product by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50023464(CHEMBL3326521)
Affinity DataKi:  360nMAssay Description:Inhibition of recombinant human CYP19A1 assessed as inhibition of DBF conversion to fluorescein by-product by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM31768(CHEMBL295698 | Ketoconazole | Nizoral | Panfungol)
Affinity DataKi:  398nMAssay Description:Inhibition of human recombinant aromatase assessed as conversion of O-dibenzylfluorescein benzyl ester substrate to fluorescein byproduct by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM31768(CHEMBL295698 | Ketoconazole | Nizoral | Panfungol)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant aromatase assessed as conversion of O-dibenzylfluorescein benzyl ester substrate to fluorescein byproduct by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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