Affinity DataIC50: 0.0900nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Evaluated for binding affinity against Melanocortin-4 receptor by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: <0.400nMAssay Description:Inhibitory activity against HIV-1 Protease was determinedMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
University Of Manchester
Curated by ChEMBL
University Of Manchester
Curated by ChEMBL
Affinity DataIC50: 0.410nMAssay Description:Inhibition of human RET cytoplasmic domain (658 to 1114 residues) expressed in baculovirus system preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Evaluated for binding affinity against Melanocortin-4 receptor by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Evaluated for binding affinity against rat Melanocortin-4 receptor (rMC4R) by displacing [125I]NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.660nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
University Of Manchester
Curated by ChEMBL
University Of Manchester
Curated by ChEMBL
Affinity DataIC50: 0.75nMAssay Description:Inhibition of human RET cytoplasmic domain (658 to 1114 residues) expressed in baculovirus system preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.930nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
University Of Manchester
Curated by ChEMBL
University Of Manchester
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human RET cytoplasmic domain (658 to 1114 residues) expressed in baculovirus system preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Evaluated for binding affinity against Melanocortin-4 receptor by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Evaluated for Functional Activity at Melanocortin-4 receptor as effective concentration at 50% maximum CMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Evaluated for binding affinity against human Melanocortin-4 receptor (hMC4R) by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against HSV-2 Thymidine Kinase (HSV-2 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against HIV-1 Protease was determinedMore data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
University Of Manchester
Curated by ChEMBL
University Of Manchester
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human RET cytoplasmic domain (658 to 1114 residues) expressed in baculovirus system preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against HIV-1 Protease was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against HIV-1 Protease was determinedMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
University Of Manchester
Curated by ChEMBL
University Of Manchester
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human RET cytoplasmic domain (658 to 1114 residues) expressed in baculovirus system preincubated for 15 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Roche Discovery Welwyn
Curated by ChEMBL
Roche Discovery Welwyn
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against HSV-1 Thymidine Kinase (HSV-1 TK)More data for this Ligand-Target Pair