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Found 221 with Last Name = 'hoshi' and Initial = 'k'
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Josai University

Curated by ChEMBL
LigandPNGBDBM50568282(CHEMBL4847545)
Affinity DataKi:  1.5nMAssay Description:Mixed type inhibition of human recombinant MAO-B by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171475(CHEMBL190288 | {3-[2-(Diphenyl-ethanesulfonyl)-eth...)
Affinity DataKi:  4.30nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171478(CHEMBL190236 | {3-[2-(1,1-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50332808((8R,9S,10S,13S,14S)-10-(hydroxymethyl)-13-methyl-2...)
Affinity DataKi:  13nMAssay Description:Inhibition of 1 uM [1-beta-3H]-androstenedione binding to human placental microsome Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50332807((8R,9S,10R,13S,14S)-10,13-dimethyl-2,3,7,8,9,10,11...)
Affinity DataKi:  13nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Josai University

Curated by ChEMBL
LigandPNGBDBM50568281(CHEMBL1241163)
Affinity DataKi:  18nMAssay Description:Mixed type inhibition of human recombinant MAO-B by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50025428(10,13-Dimethyl-1,6,7,8,9,10,11,12,13,14,15,16-dode...)
Affinity DataKi:  20nMAssay Description:Binding affinity for aromatase cytochrome P45019A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171477(CHEMBL191056 | {3-[2-(1,1-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  26nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50332807((8R,9S,10R,13S,14S)-10,13-dimethyl-2,3,7,8,9,10,11...)
Affinity DataKi:  37nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171483(CHEMBL365501 | {3-[2-(Diphenyl-ethanesulfinyl)-eth...)
Affinity DataKi:  51nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039154(10,13-Dimethyl-1,2,7,8,9,10,11,12,13,14,15,16-dode...)
Affinity DataKi:  58nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171472(CHEMBL190840 | [3-[2-(1,1-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  72nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171474(CHEMBL192662 | [3-[2-(1,1-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  78nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171466(CHEMBL361939 | {3-[2-(2,2-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  80nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171466(CHEMBL361939 | {3-[2-(2,2-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  80nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171465(CHEMBL190708 | [3-(2-Benzhydrylsulfanyl-ethyl)-2-h...)
Affinity DataKi:  88nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50422015(CHEMBL2311169)
Affinity DataKi:  120nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039160(13-Methyl-1,6,7,8,9,10,11,12,13,14,15,16-dodecahyd...)
Affinity DataKi:  140nMAssay Description:Binding affinity for aromatase cytochrome P45019A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171480(CHEMBL191118 | {2-Hydroxymethyl-3-[2-(2,2,2-triflu...)
Affinity DataKi:  150nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039148(10,13-Dimethyl-1,3,4,8,9,10,11,12,13,14,15,16-dode...)
Affinity DataKi:  150nMAssay Description:Time dependent inactivation of Cytochrome P450 19A1 was obtained by kitz-wilson plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009437(10-Hydroxymethyl-13-methyl-2,3,6,7,8,9,10,11,12,13...)
Affinity DataKi:  170nMAssay Description:Inhibition of 1 uM [1-beta-3H]-androstenedione binding to human placental microsome Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171479(CHEMBL189694 | {3-[2-(1,1-Diphenyl-propylsulfanyl)...)
Affinity DataKi:  180nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039158(10,13-Dimethyl-1,8,9,10,11,12,13,14,15,16-decahydr...)
Affinity DataKi:  180nMAssay Description:Time dependent inactivation of Cytochrome P450 19A1 was obtained by kitz-wilson plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171474(CHEMBL192662 | [3-[2-(1,1-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  210nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039158(10,13-Dimethyl-1,8,9,10,11,12,13,14,15,16-decahydr...)
Affinity DataKi:  220nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009430(16-Bromo-10,13-dimethyl-1,2,3,6,7,8,9,10,11,12,13,...)
Affinity DataKi:  228nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039148(10,13-Dimethyl-1,3,4,8,9,10,11,12,13,14,15,16-dode...)
Affinity DataKi:  250nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171473(CHEMBL187758 | [3-(3-Benzhydrylsulfanyl-propyl)-be...)
Affinity DataKi:  270nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009436(Acetic acid 13-methyl-17-oxo-1,2,3,6,7,8,9,11,12,1...)
Affinity DataKi:  289nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171469(CHEMBL188384 | [3-(2-Benzhydrylsulfanyl-ethyl)-ben...)
Affinity DataKi:  310nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171484(CHEMBL188758 | {3-[3-(2,2-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  400nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171469(CHEMBL188384 | [3-(2-Benzhydrylsulfanyl-ethyl)-ben...)
Affinity DataKi:  410nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009435(10-Difluoromethyl-13-methyl-1,2,3,6,7,8,9,10,11,12...)
Affinity DataKi:  443nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009431(16-Bromo-10,13-dimethyl-1,2,3,6,7,8,9,10,11,12,13,...)
Affinity DataKi:  455nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171478(CHEMBL190236 | {3-[2-(1,1-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  530nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171482(CHEMBL190735 | {3-[2-(3,3-Diphenyl-propylsulfanyl)...)
Affinity DataKi:  560nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171477(CHEMBL191056 | {3-[2-(1,1-Diphenyl-ethylsulfanyl)-...)
Affinity DataKi:  570nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171471(CHEMBL189063 | [3-(3,3-Diphenyl-propylsulfanylmeth...)
Affinity DataKi:  580nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171464(CHEMBL187544 | [3-(2,2-Diphenyl-ethylsulfanylmethy...)
Affinity DataKi:  680nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171465(CHEMBL190708 | [3-(2-Benzhydrylsulfanyl-ethyl)-2-h...)
Affinity DataKi:  750nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171480(CHEMBL191118 | {2-Hydroxymethyl-3-[2-(2,2,2-triflu...)
Affinity DataKi:  760nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009434(10,13-Dimethyl-2,3,6,7,8,9,10,11,12,13,14,15,16,17...)
Affinity DataKi:  830nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50332833((8R,9S,10S,13S,14S)-10-(hydroxymethyl)-13-methyl-3...)
Affinity DataKi:  1.00E+3nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039151(13-Methyl-17-oxo-1,2,3,4,7,8,9,11,12,13,14,15,16,1...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity for aromatase cytochrome P45019A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039155(13-Methyl-7,17-dioxo-1,2,7,8,9,11,12,13,14,15,16,1...)
Affinity DataKi:  1.80E+3nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171475(CHEMBL190288 | {3-[2-(Diphenyl-ethanesulfonyl)-eth...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039161((S)-10,13-Dimethyl-2,7,8,9,10,11,12,13,14,15,16,17...)
Affinity DataKi:  2.00E+3nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171470(CHEMBL191162 | {3-[2-(1,1-Diphenyl-butylsulfanyl)-...)
Affinity DataKi: >2.30E+3nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039150(13-Methyl-1,3,4,8,9,10,11,12,13,14,15,16-dodecahyd...)
Affinity DataKi:  2.40E+3nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50171464(CHEMBL187544 | [3-(2,2-Diphenyl-ethylsulfanylmethy...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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