Affinity DataKi: 0.00630nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.0125nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.0136nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 0.0220nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 0.0240nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.0325nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.0333nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.0435nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.177nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.214nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.218nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(CALF)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Affinity DataKi: 0.252nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 0.257nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 0.321nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.326nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.435nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(CALF)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Affinity DataKi: 0.531nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 0.682nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 0.796nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned kappa opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(CALF)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(CALF)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned kappa opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(CALF)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned kappa opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Szeged
Curated by ChEMBL
University Of Szeged
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned delta opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned kappa opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair