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Found 88 with Last Name = 'houseman' and Initial = 'bt'
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323732(3-(2-amino-1,3-benzothiazol-6-yl)-1-{[2-(4-methylp...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81369(SW13)
Affinity DataIC50:  0.700nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323728(2-((4-amino-3-(3-fluoro-5-hydroxyphenyl)-1H-pyrazo...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323731(CHEMBL1213117 | N-(6-(4-amino-1-((2-(4-methylpiper...)
Affinity DataIC50:  1nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  3nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  3nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323732(3-(2-amino-1,3-benzothiazol-6-yl)-1-{[2-(4-methylp...)
Affinity DataIC50:  4nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81371(SW18)
Affinity DataIC50:  5nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323730(2-((4-amino-3-(3-hydroxyprop-1-ynyl)-1H-pyrazolo[3...)
Affinity DataIC50:  7nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81373(SW30)
Affinity DataIC50:  7nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50324735((5E)-5-(QUINOXALIN-6-YLMETHYLENE)-1,3-THIAZOLIDINE...)
Affinity DataIC50:  8nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81370(SW14)
Affinity DataIC50:  9nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323732(3-(2-amino-1,3-benzothiazol-6-yl)-1-{[2-(4-methylp...)
Affinity DataIC50:  9nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323729(2-((4-amino-3-(3-fluoro-4-hydroxyphenyl)-1H-pyrazo...)
Affinity DataIC50:  9nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM36411(2-((4-amino-3-(3-hydroxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50:  11nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81368(PIK90)
Affinity DataIC50:  11nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  16nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81372(SW19)
Affinity DataIC50:  16nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81368(PIK90)
Affinity DataIC50:  18nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323729(2-((4-amino-3-(3-fluoro-4-hydroxyphenyl)-1H-pyrazo...)
Affinity DataIC50:  20nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323734(3-((4-amino-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidi...)
Affinity DataIC50:  21nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81370(SW14)
Affinity DataIC50:  21nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323731(CHEMBL1213117 | N-(6-(4-amino-1-((2-(4-methylpiper...)
Affinity DataIC50:  23nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81369(SW13)
Affinity DataIC50:  33nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323728(2-((4-amino-3-(3-fluoro-5-hydroxyphenyl)-1H-pyrazo...)
Affinity DataIC50:  33nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  33nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323734(3-((4-amino-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidi...)
Affinity DataIC50:  34nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323736(2-(3-(2-methoxyphenyl)-4-oxo-3,4,5,6,7,8-hexahydro...)
Affinity DataIC50:  34nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81371(SW18)
Affinity DataIC50:  38nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323733(1-(1-METHYLETHYL)-3-(PYRIDIN-3-YLETHYNYL)-1H-PYRAZ...)
Affinity DataIC50:  40nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  44nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  49nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323733(1-(1-METHYLETHYL)-3-(PYRIDIN-3-YLETHYNYL)-1H-PYRAZ...)
Affinity DataIC50:  53nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81368(PIK90)
Affinity DataIC50:  58nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50324735((5E)-5-(QUINOXALIN-6-YLMETHYLENE)-1,3-THIAZOLIDINE...)
Affinity DataIC50:  60nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323734(3-((4-amino-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidi...)
Affinity DataIC50:  69nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  75nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323735(CHEMBL1213168 | N-(3-(3,5-dimethoxyphenylamino)qui...)
Affinity DataIC50:  90nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323733(1-(1-METHYLETHYL)-3-(PYRIDIN-3-YLETHYNYL)-1H-PYRAZ...)
Affinity DataIC50:  113nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323726(2-((6-amino-9H-purin-9-yl)methyl)-5-methyl-3-o-tol...)
Affinity DataIC50:  130nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323732(3-(2-amino-1,3-benzothiazol-6-yl)-1-{[2-(4-methylp...)
Affinity DataIC50:  137nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM36411(2-((4-amino-3-(3-hydroxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50:  162nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323727(2-((9H-purin-6-ylthio)methyl)-5-chloro-3-(2-methox...)
Affinity DataIC50:  180nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323731(CHEMBL1213117 | N-(6-(4-amino-1-((2-(4-methylpiper...)
Affinity DataIC50:  185nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50323728(2-((4-amino-3-(3-fluoro-5-hydroxyphenyl)-1H-pyrazo...)
Affinity DataIC50:  220nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81369(SW13)
Affinity DataIC50:  221nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM81367(PIK293)
Affinity DataIC50:  237nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50324735((5E)-5-(QUINOXALIN-6-YLMETHYLENE)-1,3-THIAZOLIDINE...)
Affinity DataIC50:  270nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50324735((5E)-5-(QUINOXALIN-6-YLMETHYLENE)-1,3-THIAZOLIDINE...)
Affinity DataIC50:  300nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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