TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 137nMAssay Description:Inhibition of p110alphaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 162nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of p110deltaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 185nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 221nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 237nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Medical Research Council-Laboratory Of Molecular Biology
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair