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Found 22 with Last Name = 'hu' and Initial = 'yg'
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50452815(CHEMBL2005280)
Affinity DataKi:  5.11E+3nMAssay Description:Non-competitive inhibition of NDM1 in Escherichia coli BL21 (DE3) using MEPM substrate incubated for 15 mins by UV spectroscopy based L-B plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50452814(CHEMBL4212352)
Affinity DataKi:  5.63E+3nMAssay Description:Non-competitive inhibition of NDM1 in Escherichia coli BL21 (DE3) using MEPM substrate incubated for 15 mins by UV spectroscopy based L-B plotMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50452815(CHEMBL2005280)
Affinity DataIC50:  110nMAssay Description:Inhibition of NDM1 in Escherichia coli BL21 (DE3) using MEPM substrate incubated for 15 mins by UV spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223126(P5i-7)
Affinity DataIC50:  720nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223131(2-((5-(4-methoxyphenyl)furan-2-yl)methylene)hydraz...)
Affinity DataIC50:  2.10E+3nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223136(2-((6-(4-chlorophenyl)pyridin-2-yl)methylene)hydra...)
Affinity DataIC50:  3.50E+3nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223134(2-((4′-chloro-[1,1′-biphenyl]-3-yl)met...)
Affinity DataIC50:  3.80E+3nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50452814(CHEMBL4212352)
Affinity DataIC50:  5.62E+3nMAssay Description:Inhibition of NDM1 in Escherichia coli BL21 (DE3) using MEPM substrate incubated for 15 mins by UV spectroscopyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223135(2-((5-(4-chlorophenyl)pyridin-3-yl)methylene)hydra...)
Affinity DataIC50:  6.90E+3nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223127(2-((5-phenylfuran-2-yl)methylene)hydrazinecarboxam...)
Affinity DataIC50:  1.20E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223129(2-((5-(4-fluorophenyl)furan-2-yl)methylene)hydrazi...)
Affinity DataIC50:  1.20E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223133(2-((5-(2-amino-4-chlorophenyl)furan-2-yl)methylene...)
Affinity DataIC50:  1.30E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223128(2-((5-(3-fluorophenyl)furan-2-yl)methylene)hydrazi...)
Affinity DataIC50:  1.40E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223130(2-((5-(4-nitrophenyl)furan-2-yl)methylene)hydrazin...)
Affinity DataIC50:  1.80E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223132(2-((5-(4-aminophenyl)furan-2-yl)methylene)hydrazin...)
Affinity DataIC50:  4.00E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM8460(5-{[5-(4-chlorophenyl)furan-2-yl]methylidene}-2-su...)
Affinity DataIC50:  6.70E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 8(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: >1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 7(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: >1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: >1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 3 [N508S](Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: >1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: >1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 6(Homo sapiens (Human))
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: >1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed