Affinity DataIC50: 2nMAssay Description:Inhibition of human DGAT2 expressed in Sf9 cell membranes assessed as triolein formation by LC/MS/MS analysis using oleoyl-CoA as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human DGAT2 expressed in Sf9 cell membranes assessed as triolein formation by LC/MS/MS analysis using oleoyl-CoA as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human DGAT2 expressed in Sf9 cell membranes assessed as triolein formation by LC/MS/MS analysis using oleoyl-CoA as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of SCD1 in human HepG2 cells using [1-14C]stearic acid as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of SCD1 in human HepG2 cells using [1-14C]stearic acid as substrateMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of SCD1 in human HepG2 cells using radiolabeled stearic acid as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
TargetAlpha-1,6-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of MGAT2 (unknown origin) by CPM assayMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of SCD1 in human HepG2 cells using radiolabeled stearic acid as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of SCD1 in human HepG2 cells using radiolabeled stearic acid as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of SCD1 in human HepG2 cells using radiolabeled stearic acid as substrateMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of SCD1 in human HepG2 cells using [1-14C]stearic acid as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of SCD1 in human HepG2 cells using radiolabeled stearic acid as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of SCD1 in human HepG2 cells using radiolabeled stearic acid as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of SCD1 in human HepG2 cells using [1-14C]stearic acid as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of SCD1 in human HepG2 cells using radiolabeled stearic acid as substrateMore data for this Ligand-Target Pair