Compile Data Set for Download or QSAR
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Found 585 with Last Name = 'hudson' and Initial = 's'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188823(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190927(CHEMBL214513 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190919(CHEMBL386454 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188825((S)-7-(4-chlorophenyl)-3-(6-(3-(dimethylamino)pyrr...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188826((R)-7-(4-chlorophenyl)-3-(6-(3-(dimethylamino)pyrr...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190948(CHEMBL442064 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190943(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-N-((S)-1-(...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190922(5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(tetrah...)
Affinity DataKi:  2nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190931(CHEMBL265255 | N-((S)-1-((R)-3-(cyclopentylamino)p...)
Affinity DataKi:  2nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188817(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188834(7-(4-chlorophenyl)-3-(6-(3-(dimethylamino)pyrrolid...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190941(CHEMBL387013 | N-((S)-1-((R)-3-(3-cyclohexylpropyl...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190940(CHEMBL383933 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188835(7-(4-bromophenyl)-3-(6-(3-(dimethylamino)pyrrolidi...)
Affinity DataKi:  3nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190929(5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(methyl...)
Affinity DataKi:  3nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188832(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190918(CHEMBL215067 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190925(4'-Ethyl-biphenyl-4-carboxylic acid methyl-[(S)-1-...)
Affinity DataKi:  4nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190920(4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-...)
Affinity DataKi:  4nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188820(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188839(7-(benzo[d][1,3]dioxol-5-yl)-3-(6-(3-(dimethylamin...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190947(4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190934(4'-ethyl-biphenyl-4-carboxylic acid methyl-{(S)-1-...)
Affinity DataKi:  5nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190921(CHEMBL267797 | N-((S)-1-((R)-3-(dimethylamino)pyrr...)
Affinity DataKi:  5nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50170395(Biphenyl-4-carboxylic acid [6-(3-methylamino-pyrro...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188827(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190932(4'-methoxy-2'-methyl-biphenyl-4-carboxylic acid {(...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190944(5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(methyl...)
Affinity DataKi:  6nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188840(7-(4-chloro-2-methylphenyl)-3-(6-(3-(dimethylamino...)
Affinity DataKi:  7.10nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188824(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  7.20nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190933(5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-((tetra...)
Affinity DataKi:  8nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188830(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  8.80nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188841(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  10nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188836(7-(4-chloro-3-methylphenyl)-3-(6-(3-(dimethylamino...)
Affinity DataKi:  10nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190936(5-(4-methoxyphenyl)-N-methyl-N-((S)-1-((R)-3-(tetr...)
Affinity DataKi:  10nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190938(5-(4-ethylphenyl)-N-((S)-1-((R)-3-(isopropylamino)...)
Affinity DataKi:  11nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190939(4'-ethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-...)
Affinity DataKi:  11nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188833(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  13nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190935(4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-...)
Affinity DataKi:  14nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188821(7-(2,4-dichlorophenyl)-3-(6-(3-(dimethylamino)pyrr...)
Affinity DataKi:  14nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190923(CHEMBL386969 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  16nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188828(7-(2,4-dimethoxyphenyl)-3-(6-(3-(dimethylamino)pyr...)
Affinity DataKi:  16nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190930(4'-ethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-...)
Affinity DataKi:  18nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188842(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  18nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188831(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  19nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190928(CHEMBL384234 | N-((S)-1-((R)-3-(3-cyclohexylpropyl...)
Affinity DataKi:  21nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190265(4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)...)
Affinity DataKi:  22nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188816(7-(4-chlorophenyl)-3-(6-(3-(dimethylamino)pyrrolid...)
Affinity DataKi:  24nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188837(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  24nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50046071(CHEMBL3310277)
Affinity DataKi:  25nMAssay Description:Inhibition of full-length recombinant PKCepsilon (unknown origin) using ERMRPRKRQGSVRRRV peptide substrate by coupled-enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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