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Found 263 with Last Name = 'huebner' and Initial = 'h'
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526679(CHEMBL4456301)
Affinity DataKi:  0.0730nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526681(CHEMBL4537221)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526681(CHEMBL4537221)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.960nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526679(CHEMBL4456301)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526680(CHEMBL4463925)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25746(2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-methyl-4-(trifl...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]CGP12177 from human beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25746(2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-methyl-4-(trifl...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]CGP12177 from human beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR expressed in human recombinant SH-SY5Y cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246607(CHEMBL4083241)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR expressed in human recombinant SH-SY5Y cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526684(CHEMBL4437569)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526686(CHEMBL4463246)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50448377(CHEMBL3121473)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M2 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25751(Bisoprolol | Bisoprolol fumarate | Concor | [2-hyd...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526685(CHEMBL4566666)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526685(CHEMBL4566666)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246733(CHEMBL4100938)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M1 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526690(CHEMBL4553747)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526686(CHEMBL4463246)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526680(CHEMBL4463925)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246733(CHEMBL4100938)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M3 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25756((2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylami...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526682(CHEMBL4443911)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526684(CHEMBL4437569)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25756((2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylami...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]CGP12177 from human beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526690(CHEMBL4553747)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246627(CHEMBL4065555)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M1 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526687(CHEMBL4576034)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121336(CHEMBL3622098)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246733(CHEMBL4100938)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M2 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246627(CHEMBL4065555)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M3 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526683(CHEMBL4450085)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246652(CHEMBL4102555)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M1 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246675(CHEMBL4099673)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR expressed in human recombinant SH-SY5Y cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246652(CHEMBL4102555)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M3 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM25756((2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylami...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50526688(CHEMBL4473272)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121339(CHEMBL3622095)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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