Compile Data Set for Download or QSAR
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Found 61 with Last Name = 'hyun' and Initial = 'ye'
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]I-AB-MECA from recombinant human A3AR expressed in CHO cell membranes measured after 60 mins by gamma counter analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50383373(CHEMBL592652 | GSK0660)
Affinity DataKi:  4.60nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataKi:  6.10nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataKi:  10nMAssay Description:Binding affinity to PPARalpha (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  11nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataKi:  16nMAssay Description:Binding affinity to adenosine A3 receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataKi:  18nMAssay Description:Displacement of [3H] ZM241385 from wild type human A2AAR expressed in CHO cells assessed as inhibition constant incubated for 60 mins by Cheng-Prusof...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataKi:  19nMAssay Description:Displacement of [3H] ZM241385 from human A2AAR H278A mutant expressed in CHO cells assessed as inhibition constant incubated for 60 mins by Cheng-Pru...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataKi:  22nMAssay Description:Displacement of [3H] ZM241385 from human A2AAR S227A mutant expressed in CHO cells assessed as inhibition constant incubated for 60 mins by Cheng-Pru...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataKi:  56nMAssay Description:Displacement of [3H] ZM241385 from human A2AAR S277A/H278A double mutant expressed in CHO cells assessed as inhibition constant incubated for 60 mins...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyri...)
Affinity DataKi:  70nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataKi:  80nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50103521(Actos | CHEBI:8228 | Duetact | Pioglitazone | US10...)
Affinity DataKi:  96nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50555357(CHEMBL1254751)
Affinity DataKi:  106nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50555363(CHEMBL4758410)
Affinity DataKi:  374nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataKi:  392nMAssay Description:Binding affinity to adenosine A1 receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50555361(CHEMBL4799672)
Affinity DataKi:  504nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50555358(CHEMBL1254750)
Affinity DataKi:  592nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataKi:  834nMAssay Description:Displacement of [3H]MRS1754 from A2BAR (unknown origin) expressed in HEK293 cells assessed as inhibition constant by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50594422(CHEMBL5208616)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555357(CHEMBL1254751)
Affinity DataKi:  1.23E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50555362(CHEMBL4748172)
Affinity DataKi:  1.43E+3nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50555359(CHEMBL1254667)
Affinity DataKi:  1.91E+3nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50594422(CHEMBL5208616)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  3.33E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50594423(CHEMBL5208465)
Affinity DataKi:  3.40E+3nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555363(CHEMBL4758410)
Affinity DataKi:  3.56E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555359(CHEMBL1254667)
Affinity DataKi:  3.89E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555358(CHEMBL1254750)
Affinity DataKi:  4.07E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50555363(CHEMBL4758410)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555355(CHEMBL4760772)
Affinity DataKi:  7.04E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555360(CHEMBL4740559)
Affinity DataKi:  7.30E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555361(CHEMBL4799672)
Affinity DataKi:  7.66E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555356(CHEMBL4756797)
Affinity DataKi:  7.66E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555362(CHEMBL4748172)
Affinity DataKi:  9.55E+3nMAssay Description:Binding affinity to PPAR-gamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555363(CHEMBL4758410)
Affinity DataKi:  1.19E+4nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50537761(CHEMBL4638533)
Affinity DataIC50:  360nMAssay Description:Inhibition of human placental SAH hydrolase expressed in Escherichia coli JM109 using SAH as substrate preincubated for 10 mins followed by SAH addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50405728(CHEMBL2115462)
Affinity DataIC50:  370nMAssay Description:Inhibition of human placental SAH hydrolase expressed in Escherichia coli JM109 using SAH as substrate preincubated for 10 mins followed by SAH addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50537760(CHEMBL4635734)
Affinity DataIC50:  370nMAssay Description:Inhibition of human placental SAH hydrolase expressed in Escherichia coli JM109 using SAH as substrate preincubated for 10 mins followed by SAH addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50515220(CHEMBL4544781)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of human placental SAH hydrolase expressed in Escherichia coli JM109 using SAH as substrate preincubated for 10 mins followed by SAH addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50537763(CHEMBL4644901)
Affinity DataIC50:  2.03E+3nMAssay Description:Inhibition of human placental SAH hydrolase expressed in Escherichia coli JM109 using SAH as substrate preincubated for 10 mins followed by SAH addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50537764(CHEMBL4637324)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibition of human placental SAH hydrolase expressed in Escherichia coli JM109 using SAH as substrate preincubated for 10 mins followed by SAH addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50537762(CHEMBL4640283)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human placental SAH hydrolase expressed in Escherichia coli JM109 using SAH as substrate preincubated for 10 mins followed by SAH addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50594422(CHEMBL5208616)
Affinity DataEC50:  1.88E+4nMAssay Description:Antagonist activity at PPARdelta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50555363(CHEMBL4758410)
Affinity DataEC50:  9.30E+3nMAssay Description:Antagonist activity at PPARdelta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataEC50:  8.39E+3nMAssay Description:Antagonist activity at human A2AAR S277A/H278A double mutant expressed in CHO cells assessed as inhibition of CGS21680-induced cAMP accumulation prei...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataEC50:  109nMAssay Description:Antagonist activity at human A2AAR H278A mutant A2AAR expressed in CHO cells assessed as inhibition of CGS21680-induced cAMP accumulation preincubate...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataEC50:  94nMAssay Description:Antagonist activity at human A2AAR S227A mutant expressed in CHO cells assessed as inhibition of CGS21680-induced cAMP accumulation preincubated for ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataEC50:  0.900nMAssay Description:Antagonist activity at wild type human A2AAR expressed in CHO cells assessed as inhibition of CGS21680-induced cAMP accumulation preincubated for 20 ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50595579(CHEMBL5203469)
Affinity DataKd:  2.70nMAssay Description:Displacement of [3H] ZM241385 from human A2AAR S277A/H278A double mutant expressed in CHO cells assessed as dissociation constant incubated for 60 mi...More data for this Ligand-Target Pair
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