Found 29 with Last Name = 'ioele' and Initial = 'g' 
Affinity DataKi: 4.70E+3nMAssay Description:Inhibition of bovine AChE using ACH iodide as substrate preincubated for 60 mins followed by substrate addition and measured after 1 hrs by spectroph...More data for this Ligand-Target Pair
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of HCV NS5B RNA dependent RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Binding affinity to CXCR4 in human MDA-MB-231 cells preincubated for 15 mins followed by biotinylated TN41003 addition measured after 30 mins by rhod...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at CXCR4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity to CXCR4 in human MDA-MB-231 cells preincubated for 15 mins followed by biotinylated TN41003 addition measured after 30 mins by rhod...More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Binding affinity to CXCR4 in human MDA-MB-231 cells preincubated for 15 mins followed by biotinylated TN41003 addition measured after 30 mins by rhod...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]-SDF-1alpha from CXCR4 in human MDA-MB-231 cells after 60 mins by gamma-counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at CXCR4 (unknown origin)More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Calabria
Curated by ChEMBL
University Of Calabria
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of 5-lipoxygenase in rat RBL-1 cells preincubated for 10 mins followed by [14C]arachidonic acid addition and measured after 5 mins by radi...More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of endothelial lipase in mouse cells after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of endothelial lipase in human cells after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Antagonist activity at CXCR4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:Inhibition of human recombinant MetAP2 expressed in Sf9 insect cells using MAS as substrate after 30 mins by fluorometeric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Antagonist activity at CXCR4 in human MOLT-4 cells assessed as decrease in SDF-1alpha induced cytosolic Ca2+ levels preincubated for 30 mins followed...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of cyclooxygenase-1 in rat RBL-1 cells preincubated for 10 mins followed by [14C]arachidonic acid addition and measured after 5 mins by ra...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Rattus norvegicus)
University Of Calabria
Curated by ChEMBL
University Of Calabria
Curated by ChEMBL
Affinity DataIC50: <2.00E+3nMAssay Description:Inhibition of Nav1.7 in rat dorsal root ganglions at -60 mV holding potential by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of HCV genotype 1b NS5B RNA dependent RNA polymerase expressed in Escherichia coli BL21 (DE3) using biotinylated oligo-dT12 primer as subs...More data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60E+3nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+3nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
