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Found 171 with Last Name = 'jagtap' and Initial = 'p'
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM97464(US8470800, A | US8609833, 17)
Affinity DataKi:  0.970nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99192(US8501708, 12)
Affinity DataKi:  1.72nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99205(US8501708, 29)
Affinity DataKi:  2.28nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM97465(US8470800, B | US8609833, 85)
Affinity DataKi:  2.63nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99204(US8501708, 28)
Affinity DataKi:  2.65nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99197(US8501708, 17)
Affinity DataKi:  2.79nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99193(US8501708, 13)
Affinity DataKi:  2.97nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99206(US8501708, 30)
Affinity DataKi:  3.53nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99199(US8501708, 19)
Affinity DataKi:  3.61nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99202(US8501708, 22)
Affinity DataKi:  3.68nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM108258(US8609833, 91)
Affinity DataKi:  4.05nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99210(US8501708, 34)
Affinity DataKi:  4.86nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99209(US8501708, 33)
Affinity DataKi:  5.59nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM108256(CHEMBL2205239 | US8609833, 87)
Affinity DataKi:  5.79nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99208(US8501708, 32)
Affinity DataKi:  6.06nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99207(US8501708, 31)
Affinity DataKi:  6.08nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM108257(US8609833, 88)
Affinity DataKi:  7nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM97467(US8470800, D | US8609833, 93)
Affinity DataKi:  10.6nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99203(US8501708, 23)
Affinity DataKi:  12.3nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99198(US8501708, 18)
Affinity DataKi:  12.6nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99200(US8501708, 20)
Affinity DataKi:  14.4nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141447(CHEMBL279391 | N-[6-Cyclopentylamino-9-((2R,3R,4S,...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99201(US8501708, 21)
Affinity DataKi:  28.8nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99194(US8501708, 14 | US8501708, 15)
Affinity DataKi:  29nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141452(3-Cyclopentyl-N-[6-cyclopentylamino-9-((2R,3R,4S,5...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99194(US8501708, 14 | US8501708, 15)
Affinity DataKi:  53.1nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141455(CHEMBL285251 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141453(2-Cyclohexyl-N-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-h...)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141453(2-Cyclohexyl-N-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-h...)
Affinity DataKi:  207nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM108256(CHEMBL2205239 | US8609833, 87)
Affinity DataKi:  216nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141451(CHEMBL36786 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141449(CHEMBL36789 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  342nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2(Oryctolagus cuniculus (rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99205(US8501708, 29)
Affinity DataKi:  422nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141456(CHEMBL289982 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  432nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2(Oryctolagus cuniculus (rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99192(US8501708, 12)
Affinity DataKi:  476nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM97465(US8470800, B | US8609833, 85)
Affinity DataKi:  513nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99209(US8501708, 33)
Affinity DataKi:  551nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM97464(US8470800, A | US8609833, 17)
Affinity DataKi:  704nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141450(CHEMBL36320 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  733nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM99193(US8501708, 13)
Affinity DataKi:  820nMAssay Description:The compounds were studied in binding assays to determine selectivity and potency to A1, A2a and A3 adenosine receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141455(CHEMBL285251 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM108257(US8609833, 88)
Affinity DataKi:  900nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2(Homo sapiens (Human))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM108256(CHEMBL2205239 | US8609833, 87)
Affinity DataKi:  951nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141448((2S,3S,4R,5R)-5-[6-Amino-2-(3-cyclopentyl-propiony...)
Affinity DataKi:  1.01E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM108258(US8609833, 91)
Affinity DataKi:  1.02E+3nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141451(CHEMBL36786 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141450(CHEMBL36320 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141449(CHEMBL36789 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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