TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat amygdalaMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat hipocampusMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat amygdalaMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat hipocampusMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat cortexMore data for this Ligand-Target Pair
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Activation of human GABAA alpha-2-beta-3-gamma-2L receptor expressed in Xenopus oocytes assessed as modulation of nicotine-induced current by two-ele...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 4.90E+3nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 560nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 210nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataEC50: 6.30E+3nMAssay Description:Activation of human GABAA alpha-2-beta-3-gamma-2L receptor expressed in Xenopus oocytes assessed as modulation of GABA-induced current by two-electro...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Activation of human alpha-7 nAChR expressed in Xenopus oocytes assessed as modulation of nicotine-induced current by two-electrode voltage-clamp meth...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Activation of human alpha-7 nAChR expressed in Xenopus oocytes assessed as modulation of nicotine-induced current by two-electrode voltage-clamp meth...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Activation of human alpha-7 nAChR expressed in Xenopus oocytes assessed as modulation of choline-induced current by two-electrode voltage-clamp metho...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 2.50E+3nMAssay Description:Type-1 positive allosteric modulation of human alpha7 nAChR expressed in Xenopus oocytes assessed as maximum modulation of nicotine EC5 response by t...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataEC50: 34nMAssay Description:Activity at human GABAA alpha-1-beta-2-gamma-2L expressed in Xenopus oocytes assessed as potentiation of GABA currentsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Activation of human alpha-7 nAChR expressed in Xenopus oocytes assessed as modulation of acetyl choline -induced current by two-electrode voltage-cla...More data for this Ligand-Target Pair