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Found 96 with Last Name = 'jones' and Initial = 'dg'
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataKi:  0.251nMAssay Description:Inhibition of 4 nM progesterone-stimulated transactivation of MMTV-Luc reporter in CV-1 cells expressing PR-BMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataKi:  10nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474916(CHEMBL364712)
Affinity DataKi:  20nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474916(CHEMBL364712)
Affinity DataKi:  25nMAssay Description:Inhibition of 4 nM progesterone-stimulated transactivation of MMTV-Luc reporter in CV-1 cells expressing PR-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474914(CHEMBL190198)
Affinity DataKi:  40nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474917(CHEMBL366252)
Affinity DataKi:  40nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474911(CHEMBL192314)
Affinity DataKi:  40nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474912(CHEMBL190264)
Affinity DataKi:  100nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474919(CHEMBL364924)
Affinity DataKi:  100nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474914(CHEMBL190198)
Affinity DataKi:  200nMAssay Description:Inhibition of 4 nM progesterone-stimulated transactivation of MMTV-Luc reporter in CV-1 cells expressing PR-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474915(CHEMBL190900)
Affinity DataKi:  398nMAssay Description:Inhibition of 4 nM progesterone-stimulated transactivation of MMTV-Luc reporter in CV-1 cells expressing PR-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474911(CHEMBL192314)
Affinity DataKi:  794nMAssay Description:Inhibition of 4 nM progesterone-stimulated transactivation of MMTV-Luc reporter in CV-1 cells expressing PR-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474912(CHEMBL190264)
Affinity DataKi:  1.59E+3nMAssay Description:Inhibition of 4 nM progesterone-stimulated transactivation of MMTV-Luc reporter in CV-1 cells expressing PR-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474913(CHEMBL192859)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474918(CHEMBL373299)
Affinity DataKi: <3.16E+3nMAssay Description:Inhibition of 4 nM progesterone-stimulated transactivation of MMTV-Luc reporter in CV-1 cells expressing PR-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071516(2-[4-(3,4-Dichloro-phenylsulfanyl)-butyrylamino]-i...)
Affinity DataKi:  4.00E+3nMAssay Description:Compound was tested for inhibition of human phosphomannose isomerase (PMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071531(2-[4-(2,4-Dichloro-phenoxy)-butyrylamino]-indan-2-...)
Affinity DataKi:  4.00E+3nMAssay Description:Compound was tested for inhibition of yeast phosphomannose isomerase (PMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474913(CHEMBL192859)
Affinity DataKi:  5.01E+3nMAssay Description:Inhibition of 4 nM progesterone-stimulated transactivation of MMTV-Luc reporter in CV-1 cells expressing PR-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474915(CHEMBL190900)
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50474918(CHEMBL373299)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of fluorescent ligand from binding domain of progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071516(2-[4-(3,4-Dichloro-phenylsulfanyl)-butyrylamino]-i...)
Affinity DataKi:  2.60E+4nMAssay Description:Compound was evaluated for the inhibition constant against phosphomannose isomerase enzyme of Candida albicans (CaPMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415020(CHEMBL570708)
Affinity DataIC50:  2.51nMAssay Description:Agonist activity at progesterone receptor in human T47D cell after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415018(CHEMBL569353)
Affinity DataIC50:  39.8nMAssay Description:Agonist activity at progesterone receptor in human T47D cell after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415020(CHEMBL570708)
Affinity DataIC50:  50.1nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415011(CHEMBL578413)
Affinity DataIC50:  79.4nMAssay Description:Agonist activity at progesterone receptor in human T47D cell after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415018(CHEMBL569353)
Affinity DataIC50:  158nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415011(CHEMBL578413)
Affinity DataIC50:  200nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415010(CHEMBL577997)
Affinity DataIC50:  398nMAssay Description:Agonist activity at progesterone receptor in human T47D cell after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415010(CHEMBL577997)
Affinity DataIC50:  631nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415014(CHEMBL583053)
Affinity DataIC50:  794nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415015(CHEMBL571605)
Affinity DataIC50:  794nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415017(CHEMBL568893)
Affinity DataIC50:  794nMAssay Description:Agonist activity at progesterone receptor in human T47D cell after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415016(CHEMBL570916)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415011(CHEMBL578413)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415023(CHEMBL572014)
Affinity DataIC50:  1.26E+3nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415017(CHEMBL568893)
Affinity DataIC50:  1.26E+3nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415020(CHEMBL570708)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity to androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071516(2-[4-(3,4-Dichloro-phenylsulfanyl)-butyrylamino]-i...)
Affinity DataIC50:  6.00E+3nMAssay Description:Compound was tested for percentage inhibition of phosphomannose isomerase enzyme of Candida albicans (CaPMI).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Candida albicans)
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071523(2-[4-(3,4-Dichloro-phenylsulfanyl)-butyrylamino]-i...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of phosphomannose isomerase enzyme of Candida albicans (CaPMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415019(CHEMBL569354)
Affinity DataIC50:  6.31E+3nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415011(CHEMBL578413)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415013(CHEMBL572239)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415011(CHEMBL578413)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415011(CHEMBL578413)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415012(CHEMBL576296)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415021(CHEMBL572240)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of fluormone PL RED from progesterone receptor after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415011(CHEMBL578413)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Candida albicans)
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071519(2-[4-(2,4-Dichloro-phenylsulfanyl)-butyrylamino]-i...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of phosphomannose isomerase enzyme of Candida albicans (CaPMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Candida albicans)
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071539(2-[4-(3,4-Dichloro-phenoxy)-butyrylamino]-indan-2-...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of phosphomannose isomerase enzyme of Candida albicans (CaPMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Candida albicans)
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071535(2-[4-(3,4-Dichloro-phenylamino)-butyrylamino]-inda...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of phosphomannose isomerase enzyme of Candida albicans (CaPMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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