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Found 164 with Last Name = 'juliano' and Initial = 'm'
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088653(CHEMBL274152 | N-(6-Amino-2-methyl-pyridin-3-ylmet...)
Affinity DataKi:  0.0840nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088660(CHEMBL10785 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  0.210nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088657(CHEMBL11181 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  0.240nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088659(CHEMBL10346 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  0.270nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088658(CHEMBL10800 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  0.330nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088655(CHEMBL10545 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  0.360nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088652(CHEMBL275520 | N-(6-Amino-2-methyl-pyridin-3-ylmet...)
Affinity DataKi:  0.400nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088656(CHEMBL10657 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  1.60nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088661(CHEMBL275110 | N-(6-Amino-2-methyl-pyridin-3-ylmet...)
Affinity DataKi:  36nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112584(2-(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylami...)
Affinity DataKi:  50nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50370072(CHEMBL1790422)
Affinity DataKi:  100nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112580(CHEMBL268148 | PWGF(CH2NH)WWFW)
Affinity DataKi:  200nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446220(CHEMBL3109164)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088654(CHEMBL273861 | N-(6-Amino-2-methyl-pyridin-3-ylmet...)
Affinity DataKi:  350nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446221(CHEMBL3109163)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088653(CHEMBL274152 | N-(6-Amino-2-methyl-pyridin-3-ylmet...)
Affinity DataKi:  420nMAssay Description:The compound was tested for its ability to inhibit trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112597(2-{2-[2-(2-{2-[2-[2-(2-Amino-3-carboxy-propionylam...)
Affinity DataKi:  500nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088658(CHEMBL10800 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  510nMAssay Description:The compound was tested for its ability to inhibit trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088652(CHEMBL275520 | N-(6-Amino-2-methyl-pyridin-3-ylmet...)
Affinity DataKi:  580nMAssay Description:The compound was tested for its ability to inhibit trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446218(CHEMBL3109166)
Affinity DataKi:  600nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112581(6-Amino-2-(2-{2-[2-(6-amino-2-{2-[6-amino-2-(2-ami...)
Affinity DataKi:  600nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446219(CHEMBL3109165)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088660(CHEMBL10785 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  770nMAssay Description:The compound was tested for its ability to inhibit trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088657(CHEMBL11181 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  860nMAssay Description:The compound was tested for its ability to inhibit trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Federal University of Sao Paulo

LigandPNGBDBM241952(Fukugetin)
Affinity DataKi:  1.00E+3nMAssay Description:To characterize the type and extent inhibition of papain by fukugetin, papain (0.04 nM) was incubated with four concentrations of fukugetin (1.5, 3, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112596(6-Amino-2-{2-[2-(2-{2-[2-[6-amino-2-(2-amino-3-car...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112594(CHEMBL266692 | ChaALF(CH2NH)YMYY)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446218(CHEMBL3109166)
Affinity DataKi:  1.30E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446219(CHEMBL3109165)
Affinity DataKi:  1.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088659(CHEMBL10346 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  1.50E+3nMAssay Description:The compound was tested for its ability to inhibit trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataKi:  1.60E+3nMAssay Description:Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446228(CHEMBL3109061)
Affinity DataKi:  1.70E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataKi:  1.80E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446227(CHEMBL3109056)
Affinity DataKi:  1.80E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446220(CHEMBL3109164)
Affinity DataKi:  1.90E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446224(CHEMBL3109160)
Affinity DataKi:  2.30E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446211(CHEMBL3109058)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446228(CHEMBL3109061)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446224(CHEMBL3109160)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446221(CHEMBL3109163)
Affinity DataKi:  2.80E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446211(CHEMBL3109058)
Affinity DataKi:  2.90E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataKi:  3.00E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446229(CHEMBL3109060)
Affinity DataKi:  3.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataKi:  3.60E+3nMAssay Description:Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446229(CHEMBL3109060)
Affinity DataKi:  3.80E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088656(CHEMBL10657 | N-(6-Amino-2-methyl-pyridin-3-ylmeth...)
Affinity DataKi:  4.20E+3nMAssay Description:The compound was tested for its ability to inhibit trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446230(CHEMBL3109059)
Affinity DataKi:  4.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112583(1-{2-[2-[2-(6-Amino-2-{2-[2-(2-amino-3-methyl-pent...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112579(6-Amino-2-(2-{2-[2-(6-amino-2-{2-[2-(2-amino-3-cyc...)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112591(2-(2-{2-[2-(2-{2-[2-(2-Amino-4-methylsulfanyl-buty...)
Affinity DataKi:  6.50E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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