TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 0.331nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 12.3nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 20.4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 26.3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 38.0nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 55.0nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 77.6nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 141nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 166nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 219nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 269nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 347nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 355nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 437nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 437nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 479nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 741nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 741nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 813nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 813nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 832nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 912nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 933nMAssay Description:Inhibition of human recombinant FAAH assessed as conversion of [3H]AEA to [3H]ethanolamine after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 977nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 977nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of human recombinant FAAH assessed as conversion of [3H]AEA to [3H]ethanolamine after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of human recombinant FAAH assessed as conversion of [3H]AEA to [3H]ethanolamine after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant FAAH assessed as conversion of [3H]AEA to [3H]ethanolamine after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 2.57E+3nMAssay Description:Inhibition of human recombinant FAAH assessed as conversion of [3H]AEA to [3H]ethanolamine after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human recombinant FAAH assessed as conversion of [3H]AEA to [3H]ethanolamine after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 3.72E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of human recombinant MAGL using [3H]-2-OG as substrate after 10 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain
Curated by ChEMBL
Universite Catholique De Louvain
Curated by ChEMBL
Affinity DataIC50: 4.79E+3nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair