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Found 123 with Last Name = 'kato' and Initial = 'as'
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184446(CHEMBL3823961)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184416(CHEMBL3822825)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184418(CHEMBL3822572)
Affinity DataIC50:  54nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184419(CHEMBL3823445)
Affinity DataIC50:  54nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184442(CHEMBL3823351)
Affinity DataIC50:  62nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184444(CHEMBL3823394)
Affinity DataIC50:  65nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184414(CHEMBL3823131)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184415(CHEMBL3823222)
Affinity DataIC50:  122nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227933(CHEMBL77761)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory concentration against Muscarinic acetylcholine receptor derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  140nMAssay Description:Inhibition of smooth muscle cell ACAT activity for cells stimulated by cationized LDL.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184412(CHEMBL3823274)
Affinity DataIC50:  147nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184441(CHEMBL3823817)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184412(CHEMBL3823274)
Affinity DataIC50:  222nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184413(CHEMBL3823956)
Affinity DataIC50:  230nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50:  243nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-3 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227908(CHEMBL77988)
Affinity DataIC50:  311nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227935(CHEMBL75708)
Affinity DataIC50:  330nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184413(CHEMBL3823956)
Affinity DataIC50:  353nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184414(CHEMBL3823131)
Affinity DataIC50:  360nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227908(CHEMBL77988)
Affinity DataIC50:  406nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227910(CHEMBL305937)
Affinity DataIC50:  431nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227918(CHEMBL75224)
Affinity DataIC50:  446nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227912(CHEMBL75204)
Affinity DataIC50:  484nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50:  485nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184417(CHEMBL3823247)
Affinity DataIC50:  615nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50:  623nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-4 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227931(CHEMBL76938)
Affinity DataIC50:  629nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227921(CHEMBL75709)
Affinity DataIC50:  721nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  740nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in Liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  810nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in intestinal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227943(CHEMBL76935)
Affinity DataIC50:  952nMAssay Description:In vitro inhibitory concentration against ACAT derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227909(CHEMBL307505)
Affinity DataIC50:  976nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227918(CHEMBL75224)
Affinity DataIC50:  1.08E+3nMAssay Description:In vitro inhibitory concentration against ACAT derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  1.09E+3nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in Aorta (homogenate Low-density lipoproteins (LDL)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50:  1.18E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227936(CHEMBL73918)
Affinity DataIC50:  1.31E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227936(CHEMBL73918)
Affinity DataIC50:  1.41E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227907(CHEMBL441803)
Affinity DataIC50:  1.44E+3nMAssay Description:In vitro inhibitory concentration against ACAT derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227902(CHEMBL76706)
Affinity DataIC50:  1.71E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184445(CHEMBL3824102)
Affinity DataIC50:  1.79E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227915(CHEMBL421876)
Affinity DataIC50:  1.83E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227933(CHEMBL77761)
Affinity DataIC50:  2.24E+3nMAssay Description:In vitro inhibitory concentration against Muscarinic acetylcholine receptor derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227909(CHEMBL307505)
Affinity DataIC50:  2.62E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184443(CHEMBL3824269)
Affinity DataIC50:  2.82E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227932(CHEMBL77164)
Affinity DataIC50:  2.86E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184411(CHEMBL3823441)
Affinity DataIC50:  2.97E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227937(CHEMBL76258)
Affinity DataIC50:  3.01E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227948(CHEMBL75596)
Affinity DataIC50:  3.18E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227944(CHEMBL77942)
Affinity DataIC50:  3.28E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227929(CHEMBL419639)
Affinity DataIC50:  3.54E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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