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Found 103 with Last Name = 'kazimierczuk' and Initial = 'z'
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)
Affinity DataKi:  13nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34046(iodinated benzimidazole, 9a)
Affinity DataKi:  19nM ΔG°:  -45.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  23nM ΔG°:  -45.4kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34044(iodinated benzimidazole, 7a)
Affinity DataKi:  24nM ΔG°:  -45.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)
Affinity DataKi:  24nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34051(iodinated benzimidazole, 14)
Affinity DataKi:  27nM ΔG°:  -44.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)
Affinity DataKi:  31nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)
Affinity DataKi:  37nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  43nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)
Affinity DataKi:  44nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)
Affinity DataKi:  49nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34052(iodinated benzimidazole, 15)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34054(iodinated benzimidazole, 17)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  54nM ΔG°:  -43.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)
Affinity DataKi:  55nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34055(iodinated benzimidazole, 21)
Affinity DataKi:  62nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)
Affinity DataKi:  66nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34048(iodinated benzimidazole, 11a)
Affinity DataKi:  70nM ΔG°:  -42.5kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  71nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34043(iodinated benzimidazole, 6a)
Affinity DataKi:  75nM ΔG°:  -42.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)
Affinity DataKi:  77nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  78nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  80nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359844(CHEMBL1928907)
Affinity DataKi:  83nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)
Affinity DataKi:  83nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359844(CHEMBL1928907)
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34050(iodinated benzimidazole, 13a)
Affinity DataKi:  90nM ΔG°:  -41.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359847(CHEMBL1928909)
Affinity DataKi:  93nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)
Affinity DataKi:  97nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34040(iodinated benzimidazole, 3a)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)
Affinity DataKi:  100nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)
Affinity DataKi:  106nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  106nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)
Affinity DataKi:  109nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  110nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)
Affinity DataKi:  112nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)
Affinity DataKi:  112nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)
Affinity DataKi:  116nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34049(iodinated benzimidazole, 12a)
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34047(iodinated benzimidazole, 10a)
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34056(iodinated benzimidazole, 23)
Affinity DataKi:  130nM ΔG°:  -40.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)
Affinity DataKi:  133nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)
Affinity DataKi:  137nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359847(CHEMBL1928909)
Affinity DataKi:  139nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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