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Found 335 with Last Name = 'kerwar' and Initial = 's'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282079((2R,6R)-2,6-Dibenzyl-4-hydroxy-heptanedioic acid b...)
Affinity DataKi:  3.5nMAssay Description:Compound was evaluated for its binding affinity against HIV-1 protease using [125I]-SPA (scintillation proximity assay)More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282079((2R,6R)-2,6-Dibenzyl-4-hydroxy-heptanedioic acid b...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282083((S)-2-((S)-2-{(2R,6R)-2-Benzyl-4-hydroxy-6-[(S)-1-...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282077((S)-2-((S)-2-{(2R,6R)-2-Butyl-4-hydroxy-6-[(S)-1-(...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282076((S)-2-((S)-2-{(2R,6R)-2-Benzyl-4-hydroxy-6-[(S)-1-...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282087((2R,6R)-2,6-Dibenzyl-4-hydroxy-heptanedioic acid b...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PAF-induced platelet aggregation in rabbit platelet rich plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50047776(2-{[Acetyl-(3-tert-butyl-4-tetradecyloxy-benzoyl)-...)
Affinity DataIC50:  22nMAssay Description:Inhibition of PAF-induced platelet aggregation in rabbit platelet rich plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282081((S)-2-((S)-2-{(2R,6R)-2-Benzyl-4-hydroxy-6-[(S)-1-...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282097((3S,4aS,8aS)-2-((R)-4-{(1S,2S)-1-[(1H-Benzoimidazo...)
Affinity DataIC50:  30nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282098(1-((R)-4-{(1S,2S)-1-[(1H-Benzoimidazol-2-ylmethyl)...)
Affinity DataIC50:  30nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50403198(CHEMBL2114445)
Affinity DataIC50:  30nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50403197(CHEMBL2115378)
Affinity DataIC50:  30nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM519((2S)-N-[(2S,3R)-4-[(3S,4aS,8aS)-3-(tert-butylcarba...)
Affinity DataIC50:  30nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284036((2R,6R)-2,6-Dibenzyl-4-hydroxy-heptanedioic acid b...)
Affinity DataIC50:  40nMAssay Description:Compound was tested for inhibitory activity against recombinant HIV-1 protease using 125 I-SPA (scintillation proximity assay)More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284034((2R,6R)-2,6-Dibenzyl-4-hydroxy-heptanedioic acid b...)
Affinity DataIC50:  45nMAssay Description:Compound was tested for inhibitory activity against recombinant HIV-1 protease using 125 I-SPA (scintillation proximity assay)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50047782(2-{[Acetyl-(3-methoxy-4-tetradecyloxy-benzoyl)-ami...)
Affinity DataIC50:  64nMAssay Description:Inhibition of PAF-induced platelet aggregation in rabbit platelet rich plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282103((3S,4aS,8aS)-2-((R)-4-{(1S,2S)-1-[(1H-Benzoimidazo...)
Affinity DataIC50:  70nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282092(CHEMBL412878 | Isoquinoline-3-carboxylic acid {(1S...)
Affinity DataIC50:  70nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282095(CHEMBL291155 | Quinoline-2-carboxylic acid {(1S,2S...)
Affinity DataIC50:  70nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282078((S)-2-((S)-2-{(2R,6R)-2-Butyl-4-hydroxy-6-[(S)-1-(...)
Affinity DataIC50:  75nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50138607(2-{4-[(R)-2-Hydroxy-3-(2-methyl-benzothiazol-5-ylo...)
Affinity DataIC50:  77nMAssay Description:Inhibitory activity against Palmitoyl-CoA oxidase to inhibit rat heart mitochondrial Palmitoyl-CoA oxidation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282091(1-((R)-4-{(1S,2S)-1-[(1H-Benzoimidazol-2-ylmethyl)...)
Affinity DataIC50:  80nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50006082(3-{3-[(2,5-Di-tert-butyl-4-dodecyloxy-phenoxy)-hyd...)
Affinity DataIC50:  90nMAssay Description:Inhibition of PAF induced platelet aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282085((S)-2-((S)-2-{(2R,6R)-2-Butyl-4-hydroxy-6-[(S)-1-(...)
Affinity DataIC50:  90nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50047772(CHEMBL349327 | Trifluoro-methanesulfonate2-{[acety...)
Affinity DataIC50:  100nMAssay Description:Inhibition of PAF-induced platelet aggregation in rabbit platelet rich plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50138628(2-{4-[(R)-2-Hydroxy-3-(2-methyl-benzothiazol-5-ylo...)
Affinity DataIC50:  105nMAssay Description:Inhibitory activity against Palmitoyl-CoA oxidase to inhibit rat heart mitochondrial Palmitoyl-CoA oxidation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50156430((R)-1-{(S)-4-[5-(2,4-Dichloro-phenyl)-[1,2,4]oxadi...)
Affinity DataIC50:  120nMAssay Description:Inhibition of palmitoyl-CoA oxidation in rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50156430((R)-1-{(S)-4-[5-(2,4-Dichloro-phenyl)-[1,2,4]oxadi...)
Affinity DataIC50:  120nMAssay Description:Inhibition of palmitoyl-CoA oxidation in rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50156421((R)-1-{4-[5-(2,4-Dichloro-phenyl)-[1,2,4]oxadiazol...)
Affinity DataIC50:  130nMAssay Description:Inhibition of palmitoyl-CoA oxidation in rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282099((4S,8aS)-2-((S)-4-{1-[(S,S)-(R)-2-(1H-Benzoimidazo...)
Affinity DataIC50:  130nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50006092(3-{3-[(2,6-Di-tert-butyl-4-dodecyloxy-phenoxy)-hyd...)
Affinity DataIC50:  130nMAssay Description:Inhibition of PAF induced platelet aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282100((R)-2-Benzyl-5-[(tert-butylcarbamoyl-methyl)-cyclo...)
Affinity DataIC50:  140nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50138619(2-{4-[(R)-2-Hydroxy-3-(2-methyl-benzothiazol-5-ylo...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against Palmitoyl-CoA oxidase to inhibit rat heart mitochondrial Palmitoyl-CoA oxidation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282101((3S,4aS,8aS)-2-((R)-2-Hydroxy-4-{(1S,2S)-2-methyl-...)
Affinity DataIC50:  150nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50047761(2-{[Acetyl-(3-methoxy-4-tetradecyloxy-benzoyl)-ami...)
Affinity DataIC50:  160nMAssay Description:Inhibition of PAF-induced platelet aggregation in rabbit platelet rich plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50006071(3-{3-[Hydroxy-(2-methoxy-3-octadecylcarbamoyloxy-p...)
Affinity DataIC50:  170nMAssay Description:Inhibition of PAF induced platelet aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50138602(CHEMBL152968 | N-Biphenyl-3-yl-2-{4-[(R)-2-hydroxy...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity against Palmitoyl-CoA oxidase to inhibit rat heart mitochondrial Palmitoyl-CoA oxidation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50156415((R)-1-{4-[5-(4-tert-Butyl-phenyl)-[1,2,4]oxadiazol...)
Affinity DataIC50:  180nMAssay Description:Inhibition of palmitoyl-CoA oxidation in rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50138617(2-{4-[(R)-2-Hydroxy-3-(2-methyl-benzothiazol-5-ylo...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against Palmitoyl-CoA oxidase to inhibit rat heart mitochondrial Palmitoyl-CoA oxidation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50006003(3-{3-[Hydroxy-(5-tetradecyloxy-biphenyl-2-yloxy)-p...)
Affinity DataIC50:  200nMAssay Description:Inhibition of PAF induced platelet aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50006061(3-{3-[Hydroxy-(2,3,6-trimethyl-4-tetradecyloxy-phe...)
Affinity DataIC50:  210nMAssay Description:Inhibition of PAF induced platelet aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50006076(3-(3-{[3-(3-Dodecyloxy-2-methyl-phenoxy)-2-ethoxy-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of PAF induced platelet aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50156413((R)-1-(2-Methyl-benzothiazol-5-yloxy)-3-{(S)-2-met...)
Affinity DataIC50:  250nMAssay Description:Inhibition of palmitoyl-CoA oxidation in rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50282102(1-((R)-2-Hydroxy-4-{(1S,2S)-2-methyl-1-[(pyridin-2...)
Affinity DataIC50:  250nMAssay Description:Concentration required for inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50006029(3-{3-[(2-Acetyl-4-tetradecyloxy-phenoxy)-hydroxy-p...)
Affinity DataIC50:  300nMAssay Description:Inhibition of PAF induced platelet aggregation in rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50138625(2-{4-[(R)-2-Hydroxy-3-(2-methyl-benzothiazol-5-ylo...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Palmitoyl-CoA oxidase to inhibit rat heart mitochondrial Palmitoyl-CoA oxidation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284031((2R,6R)-2,6-Dibenzyl-4-hydroxy-heptanedioic acid b...)
Affinity DataIC50:  350nMAssay Description:Compound was tested for inhibitory activity against recombinant HIV-1 protease using 125 I-SPA (scintillation proximity assay)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50138627(2-{4-[(R)-2-Hydroxy-3-(2-methyl-benzothiazol-5-ylo...)
Affinity DataIC50:  360nMAssay Description:Inhibitory activity against Palmitoyl-CoA oxidase to inhibit rat heart mitochondrial Palmitoyl-CoA oxidation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal acyl-coenzyme A oxidase 1(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50156414((R)-1-(2-Methyl-benzothiazol-5-yloxy)-3-{4-[5-(4-t...)
Affinity DataIC50:  380nMAssay Description:Inhibition of palmitoyl-CoA oxidation in rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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