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Found 9 with Last Name = 'khudeir' and Initial = 'n'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50260210(4'-O-beta-D-glucosyl-9-O-(6' '-deoxysaccharosyl)ol...)
Affinity DataKi:  26nMAssay Description:Displacement [3H]DPCPX from of human adenosine A1 receptor at high affinity state expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50260210(4'-O-beta-D-glucosyl-9-O-(6' '-deoxysaccharosyl)ol...)
Affinity DataKi:  5.28E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM10849(1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-d...)
Affinity DataKi:  2.35E+4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50260210(4'-O-beta-D-glucosyl-9-O-(6' '-deoxysaccharosyl)ol...)
Affinity DataKi:  2.36E+4nMAssay Description:Displacement [3H]DPCPX from of human adenosine A1 receptor at low affinity state expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50260210(4'-O-beta-D-glucosyl-9-O-(6' '-deoxysaccharosyl)ol...)
Affinity DataKi:  3.10E+4nMAssay Description:Displacement [3H]DPCPX from of human adenosine A1 receptor expressed in CHO cells in presence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM10849(1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-d...)
Affinity DataKi:  3.25E+4nMAssay Description:Displacement of [3H]MSX-2 from A2A receptor in rat brain striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at adenosine A1 receptor in rat cortical membrane assessed as reduction of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50260210(4'-O-beta-D-glucosyl-9-O-(6' '-deoxysaccharosyl)ol...)
Affinity DataEC50:  3.98E+3nMAssay Description:Agonist activity at adenosine A1 receptor in rat cortical membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataEC50:  16.9nMAssay Description:Agonist activity at adenosine A1 receptor in rat cortical membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed