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Found 357 with Last Name = 'kim' and Initial = 'ja'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataKi:  10nMAssay Description:Binding affinity to PPARalpha (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyri...)
Affinity DataKi:  70nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataKi:  80nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM60579((5Z)-5-(4-hydroxybenzylidene)thiazolidine-2,4-quin...)
Affinity DataKi:  374nMAssay Description:Competitive inhibition of mushroom tyrosinase using L-tyrosine as substrate at 1.25 uM by Line-Weaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM50485276(CHEMBL233375)
Affinity DataKi:  413nMAssay Description:Competitive inhibition of mushroom tyrosinase using L-tyrosine as substrate at 1.25 uM by Line-Weaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM33932(4-(3H-1,3-benzothiazol-2-ylidene)-1-cyclohexa-2,5-...)
Affinity DataKi:  567nMAssay Description:Inhibition of mushroom tyrosinase at 1.25 uM by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM50339940(4-(Benzo[d]thiazol-2-yl)benzene-1,3-diol | CHEMBL1...)
Affinity DataKi:  673nMAssay Description:Inhibition of mushroom tyrosinase at 1.25 uM by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM60579((5Z)-5-(4-hydroxybenzylidene)thiazolidine-2,4-quin...)
Affinity DataKi:  840nMAssay Description:Competitive inhibition of mushroom tyrosinase using L-tyrosine as substrate at 20 uM by Line-Weaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyungpook National University

Curated by ChEMBL
LigandPNGBDBM50537869(CHEMBL4638367)
Affinity DataKi:  920nMAssay Description:Inhibition of PTP1B (unknown origin) assessed as decrease in p-nitrophenolate formation using using pNPP as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Catholic University Of Daegu

Curated by ChEMBL
LigandPNGBDBM50092532(CHEMBL3586200)
Affinity DataKi:  990nMAssay Description:Inhibition of BChE (unknown origin) by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50594422(CHEMBL5208616)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyungpook National University

Curated by ChEMBL
LigandPNGBDBM50537867(CHEMBL4649760)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of PTP1B (unknown origin) assessed as decrease in p-nitrophenolate formation using using pNPP as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Catholic University Of Daegu

Curated by ChEMBL
LigandPNGBDBM50092540(CHEMBL3586207)
Affinity DataKi:  1.17E+3nMAssay Description:Inhibition of AChE (unknown origin) by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM50485276(CHEMBL233375)
Affinity DataKi:  1.38E+3nMAssay Description:Competitive inhibition of mushroom tyrosinase using L-tyrosine as substrate at 20 uM by Line-Weaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM33932(4-(3H-1,3-benzothiazol-2-ylidene)-1-cyclohexa-2,5-...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of mushroom tyrosinase at 20 uM by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Catholic University Of Daegu

Curated by ChEMBL
LigandPNGBDBM50092531(CHEMBL3586199)
Affinity DataKi:  2.49E+3nMAssay Description:Inhibition of AChE (unknown origin) by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50594422(CHEMBL5208616)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyungpook National University

Curated by ChEMBL
LigandPNGBDBM226157(PTP1B spring 7 (7))
Affinity DataKi:  3.00E+3nM ΔG°:  -32.8kJ/mole IC50:  4.80E+3nMpH: 6.0 T: 2°CAssay Description:In each 96-well plates (total 200 μL of volume), there were 2 mM p-NPP and PTP1B (0.05-0.1 μg) in a buffer containing 50 mM citrate (pH 6.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50594423(CHEMBL5208465)
Affinity DataKi:  3.40E+3nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555363(CHEMBL4758410)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
Catholic University Of Daegu

Curated by ChEMBL
LigandPNGBDBM50092529(CHEMBL3586197)
Affinity DataKi:  4.78E+3nMAssay Description:Inhibition of BChE (unknown origin) by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Catholic University Of Daegu

Curated by ChEMBL
LigandPNGBDBM50092533(CHEMBL3586201)
Affinity DataKi:  4.88E+3nMAssay Description:Inhibition of BChE (unknown origin) by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM50339940(4-(Benzo[d]thiazol-2-yl)benzene-1,3-diol | CHEMBL1...)
Affinity DataKi:  7.70E+3nMAssay Description:Inhibition of mushroom tyrosinase at 20 uM by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Catholic University Of Daegu

Curated by ChEMBL
LigandPNGBDBM50092532(CHEMBL3586200)
Affinity DataKi:  7.97E+3nMAssay Description:Inhibition of AChE (unknown origin) by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyungpook National University

Curated by ChEMBL
LigandPNGBDBM226153(Selaginellin U (2))
Affinity DataKi:  9.70E+3nM ΔG°:  -29.8kJ/mole IC50:  1.38E+4nMpH: 6.0 T: 2°CAssay Description:In each 96-well plates (total 200 μL of volume), there were 2 mM p-NPP and PTP1B (0.05-0.1 μg) in a buffer containing 50 mM citrate (pH 6.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyungpook National University

Curated by ChEMBL
LigandPNGBDBM226155(Selaginellin W (4))
Affinity DataKi:  1.11E+4nM ΔG°:  -29.4kJ/mole IC50:  1.46E+4nMpH: 6.0 T: 2°CAssay Description:In each 96-well plates (total 200 μL of volume), there were 2 mM p-NPP and PTP1B (0.05-0.1 μg) in a buffer containing 50 mM citrate (pH 6.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyungpook National University

Curated by ChEMBL
LigandPNGBDBM226154(Selaginellin V (3))
Affinity DataKi:  1.13E+4nM ΔG°:  -29.4kJ/mole IC50:  1.45E+4nMpH: 6.0 T: 2°CAssay Description:In each 96-well plates (total 200 μL of volume), there were 2 mM p-NPP and PTP1B (0.05-0.1 μg) in a buffer containing 50 mM citrate (pH 6.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50555363(CHEMBL4758410)
Affinity DataKi:  1.19E+4nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET based LanthaScreen competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyungpook National University

Curated by ChEMBL
LigandPNGBDBM226156(PTP1B spring 5 (5))
Affinity DataKi:  1.39E+4nM ΔG°:  -28.8kJ/mole IC50:  1.59E+4nMpH: 6.0 T: 2°CAssay Description:In each 96-well plates (total 200 μL of volume), there were 2 mM p-NPP and PTP1B (0.05-0.1 μg) in a buffer containing 50 mM citrate (pH 6.0...More data for this Ligand-Target Pair
In DepthDetails
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyungpook National University

Curated by ChEMBL
LigandPNGBDBM50093523(CHEMBL3585679 | PTP1B spring 6 (6))
Affinity DataKi:  1.45E+4nM ΔG°:  -28.7kJ/mole IC50:  1.32E+4nMpH: 6.0 T: 2°CAssay Description:In each 96-well plates (total 200 μL of volume), there were 2 mM p-NPP and PTP1B (0.05-0.1 μg) in a buffer containing 50 mM citrate (pH 6.0...More data for this Ligand-Target Pair
In DepthDetails
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Pusan National University

Curated by ChEMBL
LigandPNGBDBM50339940(4-(Benzo[d]thiazol-2-yl)benzene-1,3-diol | CHEMBL1...)
Affinity DataIC50:  10nMAssay Description:Inhibition of mushroom tyrosinase using L-tyrosine as a substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545490(CHEMBL4644839)
Affinity DataIC50:  12nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545487(CHEMBL4635915)
Affinity DataIC50:  13nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545485(CHEMBL4633775)
Affinity DataIC50:  13nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545488(CHEMBL4638530)
Affinity DataIC50:  14nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545491(CHEMBL4642853)
Affinity DataIC50:  16nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545507(CHEMBL4641173)
Affinity DataIC50:  18nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545486(CHEMBL4644651)
Affinity DataIC50:  19nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545484(CHEMBL4634040)
Affinity DataIC50:  19nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545509(CHEMBL4642364)
Affinity DataIC50:  23nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545495(CHEMBL4638065)
Affinity DataIC50:  24nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545489(CHEMBL4648894)
Affinity DataIC50:  24nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545508(CHEMBL4634273)
Affinity DataIC50:  24nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545511(CHEMBL4636907)
Affinity DataIC50:  27nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545494(CHEMBL4647752)
Affinity DataIC50:  28nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545503(CHEMBL4635745)
Affinity DataIC50:  33nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545497(CHEMBL4649017)
Affinity DataIC50:  38nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545498(CHEMBL4636693)
Affinity DataIC50:  38nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50545513(CHEMBL4638951)
Affinity DataIC50:  42nMAssay Description:Inhibition of HSP90 (unknown origin) assessed as HER2 degradation by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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