Affinity DataKi: 0.00230nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0190nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0420nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0460nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0690nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0920nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.146nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity for rat Adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.336nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Science And Technology (Ust)
Curated by ChEMBL
University Of Science And Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Binding affinity to PLK1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Korea Institute Of Science & Technology
Curated by ChEMBL
Korea Institute Of Science & Technology
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of Phosphodiesterase 5 from rat diaphragmMore data for this Ligand-Target Pair
Affinity DataKi: >5nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: >5nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Mixed/noncompetitive inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Mixed/noncompetitive inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetSialidase(Clostridium perfringens)
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 67nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor in CHO cells (hA3)More data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
TargetSialidase(Clostridium perfringens)
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
TargetSialidase(Clostridium perfringens)
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
TargetSialidase(Clostridium perfringens)
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 127nMAssay Description:Apparent binding affinity at Clostridium perfringens neuraminidase by fluorimetryMore data for this Ligand-Target Pair
TargetSialidase(Clostridium perfringens)
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Graduate School Of Gyeongsang National University
Curated by ChEMBL
Affinity DataKi: 136nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair