Affinity DataKi: 0.0851nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.145nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health
Curated by PDSP Ki Database
National Institute of Mental Health
Curated by PDSP Ki Database
Affinity DataKi: 0.151nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute of Mental Health
Curated by PDSP Ki Database
National Institute of Mental Health
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of 20 pM [125I]BH-CCK-8S binding to mouse cortical membrane Cholecystokinin 2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health
Curated by PDSP Ki Database
National Institute of Mental Health
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health
Curated by PDSP Ki Database
National Institute of Mental Health
Curated by PDSP Ki Database