TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Competitive inhibition of VEGFR2 by qPCR methodMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Competitive inhibition of recombinant GST-tagged VEGFR2 cytoplasmic domain in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]neurotensin from NTR1 in human HT29 cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human full-length ERbeta expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant COX-2 by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant COX2 by enzymatic fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human full-length ERbeta expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human full-length ERbeta expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Displacement of [3H]neurotensin from NTR1 in human HT29 cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 810nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant COX2 by enzymatic fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human full-length ERbeta expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induced...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at human full-length ERbeta expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induced...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human full-length ERbeta expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human full-length ERalpha expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induce...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant COX-2 by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Antagonist activity at human full-length ERbeta expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human recombinant COX-2 by fluorescence assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human full-length ERbeta expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induced...More data for this Ligand-Target Pair