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Found 74 with Last Name = 'kobayashi' and Initial = 'd'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50019290(CHEMBL3289390)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50377964(Cantil | Glycophenylate | MEPENZOLATE BROMIDE | Me...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50019290(CHEMBL3289390)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50019289(CHEMBL3289391)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50377964(Cantil | Glycophenylate | MEPENZOLATE BROMIDE | Me...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613945(CHEMBL5289073)
Affinity DataKi:  10nMAssay Description:Competitive inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50019289(CHEMBL3289391)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613946(5-Allyloxycoumarin | CHEMBL450963)
Affinity DataKi:  30nMAssay Description:Competitive inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613944(CHEMBL502746)
Affinity DataKi:  50nMAssay Description:Mixed type inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613947(CHEMBL448936)
Affinity DataKi:  80nMAssay Description:Competitive inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50041234(6-hydroxy-7-methoxy-5-benzofuranacrylic acid delta...)
Affinity DataKi:  90nMAssay Description:Mixed type inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613943(6-Methoxycoumarin | CHEMBL496547)
Affinity DataKi:  250nMAssay Description:Competitive inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50041234(6-hydroxy-7-methoxy-5-benzofuranacrylic acid delta...)
Affinity DataKi:  260nMAssay Description:Non competitive inhibition of CYP2A6 in human liver microsome using coumarin as substrate preincubated with NADPH for 5 mins and measured after 30 mi...More data for this Ligand-Target Pair
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613941(CHEMBL451623)
Affinity DataKi:  540nMAssay Description:Competitive inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50041234(6-hydroxy-7-methoxy-5-benzofuranacrylic acid delta...)
Affinity DataKi:  2.20E+3nMAssay Description:Competitive inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613942(8-Methoxycoumarin | CHEMBL503184)
Affinity DataKi:  4.00E+3nMAssay Description:Competitive inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50041234(6-hydroxy-7-methoxy-5-benzofuranacrylic acid delta...)
Affinity DataKi:  2.50E+4nMAssay Description:Non competitive inhibition of CYP3A4 in human liver microsome using coumarin as substrate preincubated with NADPH for 5 mins and measured after 30 mi...More data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50613946(5-Allyloxycoumarin | CHEMBL450963)
Affinity DataKi:  2.81E+4nMAssay Description:Mixed type inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
Affinity DataKi:  2.94E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50613945(CHEMBL5289073)
Affinity DataKi:  4.66E+4nMAssay Description:Mixed type inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50613947(CHEMBL448936)
Affinity DataKi:  4.24E+5nMAssay Description:Non competitive inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50613944(CHEMBL502746)
Affinity DataKi:  4.48E+5nMAssay Description:Non competitive inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAromatase(Homo sapiens (Human))
Health Sciences University Of Hokkaido

Curated by ChEMBL
LigandPNGBDBM50242734(CHEMBL4070331)
Affinity DataIC50:  29nMAssay Description:Inhibition of CYP19 in human placental microsome using [1beta-3H]-androstenedione as substrate after 15 mins in presence of NADPH by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Health Sciences University Of Hokkaido

Curated by ChEMBL
LigandPNGBDBM50242736(CHEMBL4098990)
Affinity DataIC50:  30nMAssay Description:Inhibition of CYP19 in human placental microsome using [1beta-3H]-androstenedione as substrate after 15 mins in presence of NADPH by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613945(CHEMBL5289073)
Affinity DataIC50:  40nMAssay Description:Inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAromatase(Homo sapiens (Human))
Health Sciences University Of Hokkaido

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  43nMAssay Description:Inhibition of purified HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613946(5-Allyloxycoumarin | CHEMBL450963)
Affinity DataIC50:  50nMAssay Description:Inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465930(CHEMBL4292990)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465915(CHEMBL4281315)
Affinity DataIC50:  110nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613944(CHEMBL502746)
Affinity DataIC50:  130nMAssay Description:Inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613947(CHEMBL448936)
Affinity DataIC50:  170nMAssay Description:Inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613943(6-Methoxycoumarin | CHEMBL496547)
Affinity DataIC50:  200nMAssay Description:Inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465921(CHEMBL4288439)
Affinity DataIC50:  230nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465926(CHEMBL4294614)
Affinity DataIC50:  270nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465920(CHEMBL4280558)
Affinity DataIC50:  300nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465919(CHEMBL4283397)
Affinity DataIC50:  300nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50041234(6-hydroxy-7-methoxy-5-benzofuranacrylic acid delta...)
Affinity DataIC50:  460nMAssay Description:Inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465916(CHEMBL4289183)
Affinity DataIC50:  600nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50613941(CHEMBL451623)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAromatase(Homo sapiens (Human))
Health Sciences University Of Hokkaido

Curated by ChEMBL
LigandPNGBDBM50242747(CHEMBL4078790)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of CYP19 in human placental microsome using [1beta-3H]-androstenedione as substrate after 15 mins in presence of NADPH by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Health Sciences University Of Hokkaido

Curated by ChEMBL
LigandPNGBDBM50242748(CHEMBL4103066)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of CYP19 in human placental microsome using [1beta-3H]-androstenedione as substrate after 15 mins in presence of NADPH by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465927(CHEMBL4285798)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465918(CHEMBL4282391)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465929(CHEMBL4286715)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Health Sciences University Of Hokkaido

Curated by ChEMBL
LigandPNGBDBM50242750(CHEMBL4080965)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of CYP19 in human placental microsome using [1beta-3H]-androstenedione as substrate after 15 mins in presence of NADPH by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Health Sciences University Of Hokkaido

Curated by ChEMBL
LigandPNGBDBM50242745(CHEMBL4087613)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of CYP19 in human placental microsome using [1beta-3H]-androstenedione as substrate after 15 mins in presence of NADPH by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465922(CHEMBL4277023)
Affinity DataIC50:  4.50E+3nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465931(CHEMBL4290774)
Affinity DataIC50:  6.00E+3nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465925(CHEMBL4283367)
Affinity DataIC50:  6.00E+3nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50465914(Branaplam | LMI-070 | LMI070)
Affinity DataIC50:  6.30E+3nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in CHO cell membranes after 90 mins by micro-beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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